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- Q16154408 subject Q7300121.
- Q16154408 subject Q9062291.
- Q16154408 abstract "Phosphodiesterases (PDEs) are a superfamily of enzymes. This superfamily is further classified into 11 families, PDE1 - PDE11, on the basis of regulatory properties, amino acid sequences, substrate specificities, pharmacological properties and tissue distribution. Their function is to degrade intracellular second messengers such as cyclic adenine monophosphate (cAMP) and cyclic guanosine monophosphate (cGMP) which leads to several biological processes like effect on intracellular calcium level by the Ca2+ pathway.Phosphodiesterase 5 (PDE5) is widely expressed in several tissues in the body for example brain, lung, kidney, urinary bladder, smooth muscle and platelets. It is possible to prevent cGMP hydrolysis by inhibiting PDE5 and therefore treat diseases associated with low cGMP levels, because of this, PDE5 is an ideal target for the development of inhibitors.The three major PDE5 inhibitors are sildenafil, tadalafil and vardenafil.".
- Q16154408 wikiPageExternalLink File:3D.Sild.2.png.
- Q16154408 wikiPageExternalLink File:Figure_3._PDE5_Domains.png.
- Q16154408 wikiPageExternalLink File:PDE5_SAR2.2.png.
- Q16154408 wikiPageExternalLink Figure_5._PDE5_SAR1.png.
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- Q16154408 wikiPageWikiLink Q7251477.
- Q16154408 wikiPageWikiLink Q7300121.
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- Q16154408 wikiPageWikiLink Q9062291.
- Q16154408 comment "Phosphodiesterases (PDEs) are a superfamily of enzymes. This superfamily is further classified into 11 families, PDE1 - PDE11, on the basis of regulatory properties, amino acid sequences, substrate specificities, pharmacological properties and tissue distribution.".
- Q16154408 label "Discovery and development of phosphodiesterase 5 inhibitors".