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- Irreversible_antagonist abstract "An irreversible antagonist is a type of antagonist that binds permanently to a receptor, either by forming a covalent bond to the active site, or alternatively just by binding so tightly that the rate of dissociation is effectively zero at relevant time scales. This permanently deactivates the receptor and is usually followed by rapid internalisation and recycling of the non-functional receptor protein. Irreversible enzyme inhibitors that act similarly are clinically used and include drugs such as aspirin, omeprazole and monoamine oxidase inhibitors.".
- Irreversible_antagonist wikiPageID "23590452".
- Irreversible_antagonist wikiPageLength "1144".
- Irreversible_antagonist wikiPageOutDegree "13".
- Irreversible_antagonist wikiPageRevisionID "535442892".
- Irreversible_antagonist wikiPageWikiLink Aspirin.
- Irreversible_antagonist wikiPageWikiLink Category:Receptor_antagonists.
- Irreversible_antagonist wikiPageWikiLink Covalent_bond.
- Irreversible_antagonist wikiPageWikiLink Enzyme_inhibitor.
- Irreversible_antagonist wikiPageWikiLink Irreversible_agonist.
- Irreversible_antagonist wikiPageWikiLink Monoamine_oxidase_inhibitor.
- Irreversible_antagonist wikiPageWikiLink Naloxazone.
- Irreversible_antagonist wikiPageWikiLink Omeprazole.
- Irreversible_antagonist wikiPageWikiLink Phenoxybenzamine.
- Irreversible_antagonist wikiPageWikiLink Receptor-mediated_endocytosis.
- Irreversible_antagonist wikiPageWikiLink Receptor_(biochemistry).
- Irreversible_antagonist wikiPageWikiLink Receptor_antagonist.
- Irreversible_antagonist wikiPageWikiLinkText "Irreversible antagonist".
- Irreversible_antagonist wikiPageWikiLinkText "irreversible antagonist".
- Irreversible_antagonist wikiPageWikiLinkText "irreversible".
- Irreversible_antagonist wikiPageUsesTemplate Template:Pharmacology.
- Irreversible_antagonist wikiPageUsesTemplate Template:Pharmacology-stub.
- Irreversible_antagonist wikiPageUsesTemplate Template:Reflist.
- Irreversible_antagonist subject Category:Receptor_antagonists.
- Irreversible_antagonist hypernym Antagonist.
- Irreversible_antagonist type Drug.
- Irreversible_antagonist type Antagonist.
- Irreversible_antagonist type Drug.
- Irreversible_antagonist type Concept.
- Irreversible_antagonist comment "An irreversible antagonist is a type of antagonist that binds permanently to a receptor, either by forming a covalent bond to the active site, or alternatively just by binding so tightly that the rate of dissociation is effectively zero at relevant time scales. This permanently deactivates the receptor and is usually followed by rapid internalisation and recycling of the non-functional receptor protein.".
- Irreversible_antagonist label "Irreversible antagonist".
- Irreversible_antagonist sameAs Q6073768.
- Irreversible_antagonist sameAs Antagonista_irreversible.
- Irreversible_antagonist sameAs m.06zrzc5.
- Irreversible_antagonist sameAs Необратимый_антагонист.
- Irreversible_antagonist sameAs Ireverzibilni_antagonist.
- Irreversible_antagonist sameAs Ireverzibilni_antagonist.
- Irreversible_antagonist sameAs Q6073768.
- Irreversible_antagonist sameAs 不可逆拮抗剂.
- Irreversible_antagonist wasDerivedFrom Irreversible_antagonist?oldid=535442892.
- Irreversible_antagonist isPrimaryTopicOf Irreversible_antagonist.