Matches in DBpedia 2016-04 for { <http://dbpedia.org/resource/Buprenorphine/samidorphan> ?p ?o }
- samidorphan abstract "Buprenorphine/samidorphan (developmental code name ALKS-5461) is a combination drug formulation of buprenorphine and samidorphan acting as a κ-opioid receptor (KOR) antagonist which is under development by Alkermes as an adjunct to antidepressant therapy in treatment-resistant depression (TRD). It is also under investigation by Alkermes as a treatment for cocaine dependence, which is being funded by a grant from the National Institute on Drug Abuse (NIDA).Clinical results with ALKS-5461 in Phase II have been described as \"very encouraging\", and researchers have stated that KOR antagonists including ALKS-5461 might work \"extremely well for the treatment of major depression.\" However, data from two of three core Phase III trials was recently released and revealed that ALKS-5461 was safe and well-tolerated but, disappointingly, failed to meet its primary efficacy endpoints, although some efficacy was observed. The third and final core Phase III study is currently ongoing, with results expected sometime in 2016.".
- samidorphan atcPrefix "None".
- samidorphan thumbnail Buprenorphine_and_samidorphan.svg?width=300.
- samidorphan wikiPageExternalLink 800034331.
- samidorphan wikiPageExternalLink pipeline.
- samidorphan wikiPageID "43221236".
- samidorphan wikiPageLength "32916".
- samidorphan wikiPageOutDegree "109".
- samidorphan wikiPageRevisionID "707216055".
- samidorphan wikiPageWikiLink Addiction.
- samidorphan wikiPageWikiLink Adjuvant_therapy.
- samidorphan wikiPageWikiLink Adverse_effect.
- samidorphan wikiPageWikiLink Alkermes_(company).
- samidorphan wikiPageWikiLink Analgesic.
- samidorphan wikiPageWikiLink Anhedonia.
- samidorphan wikiPageWikiLink Antidepressant.
- samidorphan wikiPageWikiLink Anxiety.
- samidorphan wikiPageWikiLink Anxiety_disorder.
- samidorphan wikiPageWikiLink Behavior.
- samidorphan wikiPageWikiLink Behavioural_despair_test.
- samidorphan wikiPageWikiLink Bipolar_disorder.
- samidorphan wikiPageWikiLink Blind_experiment.
- samidorphan wikiPageWikiLink Buprenorphine.
- samidorphan wikiPageWikiLink CERC-501.
- samidorphan wikiPageWikiLink Category:Antidepressants.
- samidorphan wikiPageWikiLink Category:Combination_drugs.
- samidorphan wikiPageWikiLink Category:Drug_rehabilitation.
- samidorphan wikiPageWikiLink Category:Kappa_antagonists.
- samidorphan wikiPageWikiLink Category:Morphinans.
- samidorphan wikiPageWikiLink Category:Semisynthetic_opioids.
- samidorphan wikiPageWikiLink Category:Synthetic_opioids.
- samidorphan wikiPageWikiLink Chronic_stress.
- samidorphan wikiPageWikiLink Clinical_trial.
- samidorphan wikiPageWikiLink Cocaine.
- samidorphan wikiPageWikiLink Combination_drug.
- samidorphan wikiPageWikiLink Conditioned_place_preference.
- samidorphan wikiPageWikiLink Constipation.
- samidorphan wikiPageWikiLink Contraindication.
- samidorphan wikiPageWikiLink Cure.
- samidorphan wikiPageWikiLink Depression_(mood).
- samidorphan wikiPageWikiLink Dizziness.
- samidorphan wikiPageWikiLink Dopamine.
- samidorphan wikiPageWikiLink Drug_interaction.
- samidorphan wikiPageWikiLink Dynorphin.
- samidorphan wikiPageWikiLink Dysphoria.
- samidorphan wikiPageWikiLink Efficacy.
- samidorphan wikiPageWikiLink Electroconvulsive_therapy.
- samidorphan wikiPageWikiLink Endogeny_(biology).
- samidorphan wikiPageWikiLink Endorphins.
- samidorphan wikiPageWikiLink Euphoria.
- samidorphan wikiPageWikiLink FDA_Fast_Track_Development_Program.
- samidorphan wikiPageWikiLink Food_and_Drug_Administration.
- samidorphan wikiPageWikiLink Gene.
- samidorphan wikiPageWikiLink Headache.
- samidorphan wikiPageWikiLink Hypothalamic–pituitary–adrenal_axis.
- samidorphan wikiPageWikiLink Investigational_New_Drug.
- samidorphan wikiPageWikiLink JDTic.
- samidorphan wikiPageWikiLink Knockout_mouse.
- samidorphan wikiPageWikiLink Ligand.
- samidorphan wikiPageWikiLink Ligand_(biochemistry).
- samidorphan wikiPageWikiLink Major_depressive_disorder.
- samidorphan wikiPageWikiLink Mania.
- samidorphan wikiPageWikiLink Mental_disorder.
- samidorphan wikiPageWikiLink Mesolimbic_pathway.
- samidorphan wikiPageWikiLink Montgomery–Åsberg_Depression_Rating_Scale.
- samidorphan wikiPageWikiLink Morphine.
- samidorphan wikiPageWikiLink National_Institute_on_Drug_Abuse.
- samidorphan wikiPageWikiLink Nausea.
- samidorphan wikiPageWikiLink Neuroplasticity.
- samidorphan wikiPageWikiLink New_drug_application.
- samidorphan wikiPageWikiLink Onset_of_action.
- samidorphan wikiPageWikiLink Opioid_antagonist.
- samidorphan wikiPageWikiLink Opioid_modulator.
- samidorphan wikiPageWikiLink Opioid_peptide.
- samidorphan wikiPageWikiLink PF-4455242.
- samidorphan wikiPageWikiLink Pain_management.
- samidorphan wikiPageWikiLink Partial_agonist.
- samidorphan wikiPageWikiLink Pentazocine.
- samidorphan wikiPageWikiLink Pharmaceutical_formulation.
- samidorphan wikiPageWikiLink Pharmacokinetics.
- samidorphan wikiPageWikiLink Phase_1.
- samidorphan wikiPageWikiLink Phases_of_clinical_research.
- samidorphan wikiPageWikiLink Physiology.
- samidorphan wikiPageWikiLink Placebo-controlled_study.
- samidorphan wikiPageWikiLink Precursor_(chemistry).
- samidorphan wikiPageWikiLink Prodynorphin.
- samidorphan wikiPageWikiLink Psychotomimetic.
- samidorphan wikiPageWikiLink Receptor_antagonist.
- samidorphan wikiPageWikiLink Samidorphan.
- samidorphan wikiPageWikiLink Sedation.
- samidorphan wikiPageWikiLink Selective_serotonin_reuptake_inhibitor.
- samidorphan wikiPageWikiLink Serotonin–norepinephrine_reuptake_inhibitor.
- samidorphan wikiPageWikiLink Stress_(biology).
- samidorphan wikiPageWikiLink Sublingual_administration.
- samidorphan wikiPageWikiLink Substance_dependence.
- samidorphan wikiPageWikiLink Therapeutic_effect.
- samidorphan wikiPageWikiLink Tolerability.
- samidorphan wikiPageWikiLink Toxicity.
- samidorphan wikiPageWikiLink Treatment-resistant_depression.
- samidorphan wikiPageWikiLink United_States.