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- H3_receptor_antagonist abstract "An H3-receptor antagonist is a classification of drugs used to block the action of histamine at the H3 receptor. Unlike the H1 and H2 receptors which have primarily peripheral actions, but cause sedation if they are blocked in the brain, H3 receptors are primarily found in the brain and are inhibitory autoreceptors located on histaminergic nerve terminals, which modulate the release of histamine. Histamine release in the brain triggers secondary release of excitatory neurotransmitters such as glutamate and acetylcholine via stimulation of H1 receptors in the cerebral cortex. Consequently unlike the H1 antagonist antihistamines which are sedating, H3 antagonists have stimulant and nootropic effects, and are being researched as potential drugs for the treatment of neurodegenerative conditions such as Alzheimer's disease.Examples of selective H3 antagonists include clobenpropit, ABT-239, ciproxifan, Conessine, A-349,821, and pitolisant".
- H3_receptor_antagonist wikiPageID "18242075".
- H3_receptor_antagonist wikiPageLength "4085".
- H3_receptor_antagonist wikiPageOutDegree "19".
- H3_receptor_antagonist wikiPageRevisionID "678841177".
- H3_receptor_antagonist wikiPageWikiLink A-349,821.
- H3_receptor_antagonist wikiPageWikiLink ABT-239.
- H3_receptor_antagonist wikiPageWikiLink Acetylcholine.
- H3_receptor_antagonist wikiPageWikiLink Alzheimers_disease.
- H3_receptor_antagonist wikiPageWikiLink Antihistamines.
- H3_receptor_antagonist wikiPageWikiLink Category:H3_receptor_antagonists.
- H3_receptor_antagonist wikiPageWikiLink Cerebral_cortex.
- H3_receptor_antagonist wikiPageWikiLink Ciproxifan.
- H3_receptor_antagonist wikiPageWikiLink Clobenpropit.
- H3_receptor_antagonist wikiPageWikiLink Conessine.
- H3_receptor_antagonist wikiPageWikiLink Glutamate.
- H3_receptor_antagonist wikiPageWikiLink Glutamic_acid.
- H3_receptor_antagonist wikiPageWikiLink Histamine.
- H3_receptor_antagonist wikiPageWikiLink Histamine_H3_receptor.
- H3_receptor_antagonist wikiPageWikiLink Histamine_antagonist.
- H3_receptor_antagonist wikiPageWikiLink Medication.
- H3_receptor_antagonist wikiPageWikiLink Nootropic.
- H3_receptor_antagonist wikiPageWikiLink Pharmaceutical_drug.
- H3_receptor_antagonist wikiPageWikiLink Pitolisant.
- H3_receptor_antagonist wikiPageWikiLink Sedation.
- H3_receptor_antagonist wikiPageWikiLink Stimulant.
- H3_receptor_antagonist wikiPageWikiLinkText "H3 receptor antagonist".
- H3_receptor_antagonist hasPhotoCollection H3_receptor_antagonist.
- H3_receptor_antagonist wikiPageUsesTemplate Template:Histaminergics.
- H3_receptor_antagonist wikiPageUsesTemplate Template:Nervous-system-drug-stub.
- H3_receptor_antagonist wikiPageUsesTemplate Template:Reflist.
- H3_receptor_antagonist subject Category:H3_receptor_antagonists.
- H3_receptor_antagonist hypernym Classification.
- H3_receptor_antagonist type Drug.
- H3_receptor_antagonist type MeanOfTransportation.
- H3_receptor_antagonist type Antagonist.
- H3_receptor_antagonist type Antihistamine.
- H3_receptor_antagonist type Drug.
- H3_receptor_antagonist type Concept.
- H3_receptor_antagonist comment "An H3-receptor antagonist is a classification of drugs used to block the action of histamine at the H3 receptor. Unlike the H1 and H2 receptors which have primarily peripheral actions, but cause sedation if they are blocked in the brain, H3 receptors are primarily found in the brain and are inhibitory autoreceptors located on histaminergic nerve terminals, which modulate the release of histamine.".
- H3_receptor_antagonist label "H3 receptor antagonist".
- H3_receptor_antagonist sameAs m.04cy798.
- H3_receptor_antagonist sameAs H3_antagonist.
- H3_receptor_antagonist sameAs Antagonist_H3_receptora.
- H3_receptor_antagonist sameAs Q5628855.
- H3_receptor_antagonist sameAs Q5628855.
- H3_receptor_antagonist wasDerivedFrom H3_receptor_antagonist?oldid=678841177.
- H3_receptor_antagonist isPrimaryTopicOf H3_receptor_antagonist.