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- Conformation_activity_relationship abstract "Conformation-activity relationship is the relationship between the biological activity and the conformation or conformational changes of a biomolecule. This terminology emphasizes the importance of dynamic conformational changes for the biological function, rather than the importance of static three-dimensional structure used in the analysis of structure activity relationships.The conformational changes usually take place during intermolecular association, such as protein–protein interaction or protein-ligand binding. A binding partner changes the conformation of a biomolecule (e.g. a protein) to enable or disable its biochemical activity. Methods for analysis of conformation activity relationship vary from in silico or using experimental methods such as X-ray crystallography and NMR where the conformation before and after activity can be compared statically or using dynamic methods such as dual polarisation interferometry or circular dichroism where the kinetics as well as degree of conformational change can be quantified.".
- Conformation_activity_relationship wikiPageID "25537414".
- Conformation_activity_relationship wikiPageLength "2518".
- Conformation_activity_relationship wikiPageOutDegree "18".
- Conformation_activity_relationship wikiPageRevisionID "454169249".
- Conformation_activity_relationship wikiPageWikiLink Binding_(molecular).
- Conformation_activity_relationship wikiPageWikiLink Biological_activity.
- Conformation_activity_relationship wikiPageWikiLink Category:Medicinal_chemistry.
- Conformation_activity_relationship wikiPageWikiLink Chemical_kinetics.
- Conformation_activity_relationship wikiPageWikiLink Chemical_structure.
- Conformation_activity_relationship wikiPageWikiLink Circular_Dichroism.
- Conformation_activity_relationship wikiPageWikiLink Circular_dichroism.
- Conformation_activity_relationship wikiPageWikiLink Conformational_change.
- Conformation_activity_relationship wikiPageWikiLink Dual-polarization_interferometry.
- Conformation_activity_relationship wikiPageWikiLink Dual_polarisation_interferometry.
- Conformation_activity_relationship wikiPageWikiLink In_silico.
- Conformation_activity_relationship wikiPageWikiLink Molecular_binding.
- Conformation_activity_relationship wikiPageWikiLink NMR.
- Conformation_activity_relationship wikiPageWikiLink Nuclear_magnetic_resonance.
- Conformation_activity_relationship wikiPageWikiLink Protein_ligand.
- Conformation_activity_relationship wikiPageWikiLink Protein–protein_interaction.
- Conformation_activity_relationship wikiPageWikiLink Structure_activity_relationship.
- Conformation_activity_relationship wikiPageWikiLink Structure–activity_relationship.
- Conformation_activity_relationship wikiPageWikiLink X-ray_crystallography.
- Conformation_activity_relationship wikiPageWikiLinkText "Conformation activity relationship".
- Conformation_activity_relationship wikiPageWikiLinkText "conformation activity relationship".
- Conformation_activity_relationship wikiPageWikiLinkText "conformation".
- Conformation_activity_relationship wikiPageWikiLinkText "conformational".
- Conformation_activity_relationship hasPhotoCollection Conformation_activity_relationship.
- Conformation_activity_relationship wikiPageUsesTemplate Template:Reflist.
- Conformation_activity_relationship subject Category:Medicinal_chemistry.
- Conformation_activity_relationship hypernym Relationship.
- Conformation_activity_relationship type Person.
- Conformation_activity_relationship type Science.
- Conformation_activity_relationship comment "Conformation-activity relationship is the relationship between the biological activity and the conformation or conformational changes of a biomolecule.".
- Conformation_activity_relationship label "Conformation activity relationship".
- Conformation_activity_relationship sameAs m.09rw_m2.
- Conformation_activity_relationship sameAs Q5160263.
- Conformation_activity_relationship sameAs Q5160263.
- Conformation_activity_relationship wasDerivedFrom Conformation_activity_relationship?oldid=454169249.
- Conformation_activity_relationship isPrimaryTopicOf Conformation_activity_relationship.