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- Q433807 subject Q8390819.
- Q433807 abstract "An orexigenic, or appetite stimulant, is a drug, hormone, or compound that increases appetite. This can be a naturally occurring neuropeptide hormone such as ghrelin, orexin or neuropeptide Y, or a medication which increases hunger and therefore enhances food consumption. Usually appetite enhancement is considered an undesirable side effect of certain drugs as it leads to unwanted weight gain, but sometimes it can be beneficial and a drug may be prescribed solely for this purpose, especially when the patient is suffering from severe appetite loss or muscle wasting due to cystic fibrosis, anorexia, old age, cancer or AIDS. There are several widely used drugs which can cause a boost in appetite, including tricyclic antidepressants (TCAs), tetracyclic antidepressants, natural or synthetic cannabinoids, first-generation antihistamines, most antipsychotics and many steroid hormones.Agents with orexigenic effects include the following: 5-HT2C receptor antagonists/inverse agonists — mirtazapine, olanzapine, quetiapine, amitriptyline, cyproheptadine H1 receptor antagonists/inverse agonists — mirtazapine, olanzapine, quetiapine, amitriptyline, cyproheptadine Dopamine antagonists — haloperidol, chlorpromazine, olanzapine, risperidone, quetiapine Adrenergic antagonists — carvedilol, propranolol; α2-adrenergic antagonists — mirtazapine; α2-adrenergic agonists – clonidine CB1 receptor agonists (cannabinoids — THC/dronabinol (a component of Cannabis), nabilone Corticosteroids — dexamethasone, prednisone, hydrocortisone Certain pregnene steroids — megestrol acetate, medroxyprogesterone acetate Anabolic steroids — oxandrolone, nandrolone, testosterone Sulfonylurea antidiabetic drugs such as glibenclamide, chlorpropamide and tolbutamide Mood stabilisers such as lithium Some anti-epileptic drugs such as valproate, carbamazepine and gabapentin α2δ VDCC ligands — pregabalin Ghrelin receptor agonists such as anamorelin, GHRP-6, ibutamoren, ipamorelin, and pralmorelin MC4 receptor antagonists Insulin Sugars such as fructose↑ ↑ ↑ ↑ ↑ ↑ ↑ ↑ ↑ ↑ ↑ ↑ ↑".
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- Q433807 wikiPageWikiLink Q8390819.
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- Q433807 comment "An orexigenic, or appetite stimulant, is a drug, hormone, or compound that increases appetite. This can be a naturally occurring neuropeptide hormone such as ghrelin, orexin or neuropeptide Y, or a medication which increases hunger and therefore enhances food consumption.".
- Q433807 label "Orexigenic".