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- Tyrosine-kinase_inhibitor abstract "A tyrosine kinase inhibitor (TKI) is a pharmaceutical drug that inhibits tyrosine kinases. Tyrosine kinases are enzymes responsible for the activation of many proteins by signal transduction cascades. The proteins are activated by adding a phosphate group to the protein (phosphorylation), a step that TKIs inhibit. TKIs are typically used as anticancer drugs. For example, they have substantially improved outcomes in chronic myelogenous leukemia.They are also called tyrphostins, the short name for “tyrosine phosphorylation inhibitor”, originally coined in a 1988 publication, which was the first description of compounds inhibiting the catalytic activity of the epidermal growth factor receptor (EGFR).The 1988 study was the first demonstration of a systematic search and discovery of small-molecular-weight inhibitors of tyrosine phosphorylation, which do not inhibit protein kinases that phosphorylate serine or threonine residues and can discriminate between the kinase domains of the EGFR and that of the insulin receptor. It was further shown that in spite of the conservation of the tyrosine-kinase domains one can design and synthesize tyrphostins that discriminate between even closely related protein tyrosine kinases such as EGFR and its close relative HER2.".
- Tyrosine-kinase_inhibitor thumbnail 3CS9_Abl1_Nilotinib.png?width=300.
- Tyrosine-kinase_inhibitor wikiPageID "27237636".
- Tyrosine-kinase_inhibitor wikiPageLength "6695".
- Tyrosine-kinase_inhibitor wikiPageOutDegree "42".
- Tyrosine-kinase_inhibitor wikiPageRevisionID "682742966".
- Tyrosine-kinase_inhibitor wikiPageWikiLink Adenosine_triphosphate.
- Tyrosine-kinase_inhibitor wikiPageWikiLink Alaska.
- Tyrosine-kinase_inhibitor wikiPageWikiLink Allosteric_regulation.
- Tyrosine-kinase_inhibitor wikiPageWikiLink Bcr-Abl_tyrosine-kinase_inhibitor.
- Tyrosine-kinase_inhibitor wikiPageWikiLink Catalysis.
- Tyrosine-kinase_inhibitor wikiPageWikiLink Category:Tyrosine_kinase_inhibitors.
- Tyrosine-kinase_inhibitor wikiPageWikiLink Cdc37.
- Tyrosine-kinase_inhibitor wikiPageWikiLink Chronic_myelogenous_leukemia.
- Tyrosine-kinase_inhibitor wikiPageWikiLink Conformational_change.
- Tyrosine-kinase_inhibitor wikiPageWikiLink Enzyme.
- Tyrosine-kinase_inhibitor wikiPageWikiLink Enzyme_inhibitor.
- Tyrosine-kinase_inhibitor wikiPageWikiLink Epidermal_growth_factor_receptor.
- Tyrosine-kinase_inhibitor wikiPageWikiLink Erlotinib.
- Tyrosine-kinase_inhibitor wikiPageWikiLink Fibroblast_growth_factor.
- Tyrosine-kinase_inhibitor wikiPageWikiLink Gefitinib.
- Tyrosine-kinase_inhibitor wikiPageWikiLink neu.
- Tyrosine-kinase_inhibitor wikiPageWikiLink Hsp90.
- Tyrosine-kinase_inhibitor wikiPageWikiLink Imatinib.
- Tyrosine-kinase_inhibitor wikiPageWikiLink Insulin_receptor.
- Tyrosine-kinase_inhibitor wikiPageWikiLink Leukemia.
- Tyrosine-kinase_inhibitor wikiPageWikiLink McKinney,_Texas.
- Tyrosine-kinase_inhibitor wikiPageWikiLink Neoplasm.
- Tyrosine-kinase_inhibitor wikiPageWikiLink Pharmaceutical_drug.
- Tyrosine-kinase_inhibitor wikiPageWikiLink Phosphate.
- Tyrosine-kinase_inhibitor wikiPageWikiLink Phosphorylation.
- Tyrosine-kinase_inhibitor wikiPageWikiLink Platelet-derived_growth_factor.
- Tyrosine-kinase_inhibitor wikiPageWikiLink Protein_kinase.
- Tyrosine-kinase_inhibitor wikiPageWikiLink Protein_kinase_inhibitor.
- Tyrosine-kinase_inhibitor wikiPageWikiLink Serine.
- Tyrosine-kinase_inhibitor wikiPageWikiLink Signal_transduction.
- Tyrosine-kinase_inhibitor wikiPageWikiLink Substrate_(chemistry).
- Tyrosine-kinase_inhibitor wikiPageWikiLink Sunitinib.
- Tyrosine-kinase_inhibitor wikiPageWikiLink Threonine.
- Tyrosine-kinase_inhibitor wikiPageWikiLink Tyrosine.
- Tyrosine-kinase_inhibitor wikiPageWikiLink Tyrosine_kinase.
- Tyrosine-kinase_inhibitor wikiPageWikiLink Ubiquitin.
- Tyrosine-kinase_inhibitor wikiPageWikiLink VEGF_receptors.
- Tyrosine-kinase_inhibitor wikiPageWikiLink Vascular_endothelial_growth_factor.
- Tyrosine-kinase_inhibitor wikiPageWikiLink File:3CS9_Abl1_Nilotinib.png.
- Tyrosine-kinase_inhibitor wikiPageWikiLinkText "Tyrosine-kinase inhibitor".
- Tyrosine-kinase_inhibitor wikiPageWikiLinkText "inhibitor of the kinase enzymes".
- Tyrosine-kinase_inhibitor wikiPageWikiLinkText "inhibitor of the tyrosine kinases".
- Tyrosine-kinase_inhibitor wikiPageWikiLinkText "tyrosine kinase inhibitor".
- Tyrosine-kinase_inhibitor wikiPageWikiLinkText "tyrosine kinase inhibitors".
- Tyrosine-kinase_inhibitor wikiPageWikiLinkText "tyrosine-kinase inhibitor".
- Tyrosine-kinase_inhibitor wikiPageUsesTemplate Template:Enzyme_inhibition.
- Tyrosine-kinase_inhibitor wikiPageUsesTemplate Template:Extracellular_chemotherapeutic_agents.
- Tyrosine-kinase_inhibitor wikiPageUsesTemplate Template:Redirect.
- Tyrosine-kinase_inhibitor wikiPageUsesTemplate Template:Reflist.
- Tyrosine-kinase_inhibitor subject Category:Tyrosine_kinase_inhibitors.
- Tyrosine-kinase_inhibitor hypernym Drug.
- Tyrosine-kinase_inhibitor type Drug.
- Tyrosine-kinase_inhibitor type Drug.
- Tyrosine-kinase_inhibitor type Inhibitor.
- Tyrosine-kinase_inhibitor type Redirect.
- Tyrosine-kinase_inhibitor comment "A tyrosine kinase inhibitor (TKI) is a pharmaceutical drug that inhibits tyrosine kinases. Tyrosine kinases are enzymes responsible for the activation of many proteins by signal transduction cascades. The proteins are activated by adding a phosphate group to the protein (phosphorylation), a step that TKIs inhibit. TKIs are typically used as anticancer drugs.".
- Tyrosine-kinase_inhibitor label "Tyrosine-kinase inhibitor".
- Tyrosine-kinase_inhibitor sameAs Q906415.
- Tyrosine-kinase_inhibitor sameAs مثبط_التيروسين_كيناز.
- Tyrosine-kinase_inhibitor sameAs Tyrosinkinase-Inhibitor.
- Tyrosine-kinase_inhibitor sameAs Inhibidor_de_la_tirosina_quinasa.
- Tyrosine-kinase_inhibitor sameAs m.0bwk09d.
- Tyrosine-kinase_inhibitor sameAs Q906415.
- Tyrosine-kinase_inhibitor wasDerivedFrom Tyrosine-kinase_inhibitor?oldid=682742966.
- Tyrosine-kinase_inhibitor depiction 3CS9_Abl1_Nilotinib.png.
- Tyrosine-kinase_inhibitor isPrimaryTopicOf Tyrosine-kinase_inhibitor.