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- Topoisomerase_inhibitor abstract "Topoisomerase inhibitors are agents designed to interfere with the action of topoisomerase enzymes (topoisomerase I and II), which are enzymes that control the changes in DNA structure by catalyzing the breaking and rejoining of the phosphodiester backbone of DNA strands during the normal cell cycle.In recent years, topoisomerases have become popular targets for cancer chemotherapy treatments. It is thought that topoisomerase inhibitors block the ligation step of the cell cycle, generating single and double stranded breaks that harm the integrity of the genome. Introduction of these breaks subsequently leads to apoptosis and cell death.Topoisomerase inhibitors can also function as antibacterial agents. Quinolones (including nalidixic acid and ciprofloxacin) have this function. Quinolones bind to these enzymes and prevent them from decatenation replicating DNA.".
- Topoisomerase_inhibitor wikiPageExternalLink NCT01051635.
- Topoisomerase_inhibitor wikiPageID "6688255".
- Topoisomerase_inhibitor wikiPageLength "27276".
- Topoisomerase_inhibitor wikiPageOutDegree "49".
- Topoisomerase_inhibitor wikiPageRevisionID "704358331".
- Topoisomerase_inhibitor wikiPageWikiLink Amsacrine.
- Topoisomerase_inhibitor wikiPageWikiLink Antibiotics.
- Topoisomerase_inhibitor wikiPageWikiLink Aurintricarboxylic_acid.
- Topoisomerase_inhibitor wikiPageWikiLink Camptothecin.
- Topoisomerase_inhibitor wikiPageWikiLink Cancer.
- Topoisomerase_inhibitor wikiPageWikiLink Cannabidiol.
- Topoisomerase_inhibitor wikiPageWikiLink Category:Antibiotics.
- Topoisomerase_inhibitor wikiPageWikiLink Category:Topoisomerase_inhibitors.
- Topoisomerase_inhibitor wikiPageWikiLink Cell_cycle.
- Topoisomerase_inhibitor wikiPageWikiLink Ciprofloxacin.
- Topoisomerase_inhibitor wikiPageWikiLink DNA.
- Topoisomerase_inhibitor wikiPageWikiLink DNA_gyrase.
- Topoisomerase_inhibitor wikiPageWikiLink DNA_ligase.
- Topoisomerase_inhibitor wikiPageWikiLink Daunorubicin.
- Topoisomerase_inhibitor wikiPageWikiLink Doxorubicin.
- Topoisomerase_inhibitor wikiPageWikiLink Ellipticines.
- Topoisomerase_inhibitor wikiPageWikiLink Enzyme.
- Topoisomerase_inhibitor wikiPageWikiLink Enzyme_catalysis.
- Topoisomerase_inhibitor wikiPageWikiLink Epigallocatechin_gallate.
- Topoisomerase_inhibitor wikiPageWikiLink Etoposide.
- Topoisomerase_inhibitor wikiPageWikiLink Genistein.
- Topoisomerase_inhibitor wikiPageWikiLink HU-331.
- Topoisomerase_inhibitor wikiPageWikiLink ICRF_193.
- Topoisomerase_inhibitor wikiPageWikiLink Irinotecan.
- Topoisomerase_inhibitor wikiPageWikiLink Lamellarin_D.
- Topoisomerase_inhibitor wikiPageWikiLink Mitoxantrone.
- Topoisomerase_inhibitor wikiPageWikiLink Nalidixic_acid.
- Topoisomerase_inhibitor wikiPageWikiLink Neoplasm.
- Topoisomerase_inhibitor wikiPageWikiLink Phenols.
- Topoisomerase_inhibitor wikiPageWikiLink Phosphodiester_bond.
- Topoisomerase_inhibitor wikiPageWikiLink Phytoalexin.
- Topoisomerase_inhibitor wikiPageWikiLink Polyphenol.
- Topoisomerase_inhibitor wikiPageWikiLink Quercetin.
- Topoisomerase_inhibitor wikiPageWikiLink Quinolone.
- Topoisomerase_inhibitor wikiPageWikiLink Resveratrol.
- Topoisomerase_inhibitor wikiPageWikiLink Tea.
- Topoisomerase_inhibitor wikiPageWikiLink Teniposide.
- Topoisomerase_inhibitor wikiPageWikiLink Topoisomerase.
- Topoisomerase_inhibitor wikiPageWikiLink Topotecan.
- Topoisomerase_inhibitor wikiPageWikiLink Type_II_topoisomerase.
- Topoisomerase_inhibitor wikiPageWikiLink Type_I_topoisomerase.
- Topoisomerase_inhibitor wikiPageWikiLink Wikt:decatenation.
- Topoisomerase_inhibitor wikiPageWikiLinkText "Topoisomerase inhibitor".
- Topoisomerase_inhibitor wikiPageWikiLinkText "inhibitor".
- Topoisomerase_inhibitor wikiPageWikiLinkText "inhibitors".
- Topoisomerase_inhibitor wikiPageWikiLinkText "topoisomerase I inhibitors".
- Topoisomerase_inhibitor wikiPageWikiLinkText "topoisomerase inhibitor".
- Topoisomerase_inhibitor wikiPageWikiLinkText "topoisomerase type II inhibitor".
- Topoisomerase_inhibitor wikiPageUsesTemplate Template:Chemotherapeutic_agents.
- Topoisomerase_inhibitor wikiPageUsesTemplate Template:Cite_journal.
- Topoisomerase_inhibitor wikiPageUsesTemplate Template:QuinoloneAntiBiotics.
- Topoisomerase_inhibitor wikiPageUsesTemplate Template:Refimprove.
- Topoisomerase_inhibitor wikiPageUsesTemplate Template:Reflist.
- Topoisomerase_inhibitor subject Category:Antibiotics.
- Topoisomerase_inhibitor subject Category:Topoisomerase_inhibitors.
- Topoisomerase_inhibitor hypernym Agents.
- Topoisomerase_inhibitor type Inhibitor.
- Topoisomerase_inhibitor type Product.
- Topoisomerase_inhibitor comment "Topoisomerase inhibitors are agents designed to interfere with the action of topoisomerase enzymes (topoisomerase I and II), which are enzymes that control the changes in DNA structure by catalyzing the breaking and rejoining of the phosphodiester backbone of DNA strands during the normal cell cycle.In recent years, topoisomerases have become popular targets for cancer chemotherapy treatments.".
- Topoisomerase_inhibitor label "Topoisomerase inhibitor".
- Topoisomerase_inhibitor sameAs Q281044.
- Topoisomerase_inhibitor sameAs Inhibiteur_de_topoisomérase.
- Topoisomerase_inhibitor sameAs m.0ghbrm.
- Topoisomerase_inhibitor sameAs Inhibitori_topoizomeraze.
- Topoisomerase_inhibitor sameAs Inhibitori_topoizomeraze.
- Topoisomerase_inhibitor sameAs Q281044.
- Topoisomerase_inhibitor wasDerivedFrom Topoisomerase_inhibitor?oldid=704358331.
- Topoisomerase_inhibitor isPrimaryTopicOf Topoisomerase_inhibitor.