Matches in DBpedia 2016-04 for { <http://dbpedia.org/resource/Selective_glucocorticoid_receptor_modulator> ?p ?o }
- Selective_glucocorticoid_receptor_modulator abstract "Selective glucocorticoid receptor modulators (SEGRMs) and selective glucocorticoid receptor agonists (SEGRAs) formerly known as dissociated glucocorticoid receptor agonists (DIGRAs) are a class of experimental drugs designed to share many of the desirable anti-inflammatory, immunosuppressive, or anticancer properties of classical glucocorticoid drugs but with fewer side effects such as skin atrophy. Although preclinical evidence on SEGRAMs’ anti-inflammatory effects are culminating, currently, the efficacy of these SEGRAMs on cancer are largely unknown.Selective glucocorticoid receptor agonists (SEGRAs) are historically and typically steroidal in structure while selective glucocorticoid receptor modulators (SEGRMs) are typically non-steroidal. The combined abbreviation of selective glucocorticoid receptor agonist and modulator is SEGRAM. A number of such ligands have been developed and are being evaluated in preclinical and clinical testing.SEGRAMs achieve their selectivity by triggering only a subset the glucocorticoid receptor mechanisms of action.".
- Selective_glucocorticoid_receptor_modulator thumbnail Mapracorat_skeletal.svg?width=300.
- Selective_glucocorticoid_receptor_modulator wikiPageID "20679814".
- Selective_glucocorticoid_receptor_modulator wikiPageLength "23604".
- Selective_glucocorticoid_receptor_modulator wikiPageOutDegree "87".
- Selective_glucocorticoid_receptor_modulator wikiPageRevisionID "707773134".
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink AP-1_transcription_factor.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Angiotensin-converting_enzyme.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Annexin_A1.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Anti-inflammatory.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Anticarcinogen.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Asthma.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Asymmetric_carbon.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Atopic_dermatitis.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Atrophoderma.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Bausch_&_Lomb.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Bayer_HealthCare_Pharmaceuticals.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Blind_experiment.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Blood_sugar.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Cahn–Ingold–Prelog_priority_rules.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Cataract.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Category:Anti-inflammatory_agents.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Category:Immunosuppressants.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Cell_nucleus.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Colitis.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Conformational_change.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Cyclooxygenase.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Cytosol.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink DNA.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink DUSP1.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Dagrocorat.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Dermatology.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Dexamethasone.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Diabetes_mellitus.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Edema.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Eye_disease.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink File:SEGRAM_basic_mechanism.tif.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Fosdagrocorat.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Glaucoma.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Glucocorticoid.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Glucocorticoid_receptor.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Heat_shock_protein.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Hormone_response_element.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink ICAM-1.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Immunophilins.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Immunosuppression.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Infection.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Intendis.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Interleukin_6.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Leukemia.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Mapracorat.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Messenger_RNA.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Metabolism.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Monomer.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink NF-κB.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Neprilysin.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Nitric_oxide_synthase.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Ophthalmology.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Osteoporosis.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Peroxidase.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Pfizer.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Phospholipase_A2.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Point_mutation.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Prednisolone.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Prodrug.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Prostaglandin_E2.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Prostate_cancer.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Protein.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Protein_dimer.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Protein_targeting.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Rheumatoid_arthritis.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Selective_androgen_receptor_modulator.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Selective_estrogen_receptor_modulator.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Selective_progesterone_receptor_modulator.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Selective_receptor_modulator.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Signal_transduction.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Steroid.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Suspension_(chemistry).
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink TSC22D3.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Topical_medication.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Transactivation.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Transforming_growth_factor_beta.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Transrepression.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink Tumor_necrosis_factors.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink File:A_276575_structure.svg.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink File:Octahydrophenanthrene-2,7-diol_SEGRA.svg.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink File:RU_24858_skeletal.svg.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLink File:Trifluoroisopropanolamine_SEGRA.svg.
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLinkText "SGRM".
- Selective_glucocorticoid_receptor_modulator wikiPageWikiLinkText "Selective glucocorticoid receptor modulator".
- Selective_glucocorticoid_receptor_modulator alt "Mapracorat".
- Selective_glucocorticoid_receptor_modulator biologicalTarget Glucocorticoid_receptor.
- Selective_glucocorticoid_receptor_modulator caption "Mapracorat, one of the furthest developed SEGRAs".
- Selective_glucocorticoid_receptor_modulator use "Potentially atopic dermatitis, glaucoma, cataract, and eye infections".
- Selective_glucocorticoid_receptor_modulator wikiPageUsesTemplate Template:Commons_category.
- Selective_glucocorticoid_receptor_modulator wikiPageUsesTemplate Template:Corticosteroids.
- Selective_glucocorticoid_receptor_modulator wikiPageUsesTemplate Template:Glucocorticoids.
- Selective_glucocorticoid_receptor_modulator wikiPageUsesTemplate Template:Good_article.
- Selective_glucocorticoid_receptor_modulator wikiPageUsesTemplate Template:Infobox_drug_class.
- Selective_glucocorticoid_receptor_modulator wikiPageUsesTemplate Template:Redirect.