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- Pyruvate_dehydrogenase_kinase abstract "Pyruvate dehydrogenase kinase (also pyruvate dehydrogenase complex kinase, PDC kinase, or PDK; EC 2.7.11.2) is a kinase enzyme which acts to inactivate the enzyme pyruvate dehydrogenase by phosphorylating it using ATP. PDK thus participates in the regulation of the pyruvate dehydrogenase complex of which pyruvate dehydrogenase is the first component. Both PDK and the pyruvate dehydrogenase complex are located in the mitochondrial matrix of eukaryotes. The complex acts to convert pyruvate (a product of glycolysis in the cytosol) to acetyl-coA, which is then oxidized in the mitochondria to produce energy, in the citric acid cycle. By downregulating the activity of this complex, PDK will decrease the oxidation of pyruvate in mitochondria and increase the conversion of pyruvate to lactate in the cytosol.The opposite action of PDK, namely the dephosphorylation and activation of pyruvate dehydrogenase, is catalyzed by a phosphoprotein phosphatase called pyruvate dehydrogenase phosphatase.(Pyruvate dehydrogenase kinase should not be confused with Phosphoinositide-dependent kinase-1, which is also sometimes known as \"PDK1\".)".
- Pyruvate_dehydrogenase_kinase ecNumber "2.7.11.2".
- Pyruvate_dehydrogenase_kinase thumbnail Pyruvate_dehydrogenase_phosphorylation_sites.png?width=300.
- Pyruvate_dehydrogenase_kinase wikiPageID "9498847".
- Pyruvate_dehydrogenase_kinase wikiPageLength "13670".
- Pyruvate_dehydrogenase_kinase wikiPageOutDegree "55".
- Pyruvate_dehydrogenase_kinase wikiPageRevisionID "705521765".
- Pyruvate_dehydrogenase_kinase wikiPageWikiLink Acetyl-CoA.
- Pyruvate_dehydrogenase_kinase wikiPageWikiLink Acetylation.
- Pyruvate_dehydrogenase_kinase wikiPageWikiLink Adenosine_diphosphate.
- Pyruvate_dehydrogenase_kinase wikiPageWikiLink Adenosine_triphosphate.
- Pyruvate_dehydrogenase_kinase wikiPageWikiLink Amino_acid.
- Pyruvate_dehydrogenase_kinase wikiPageWikiLink Apoptosis.
- Pyruvate_dehydrogenase_kinase wikiPageWikiLink Category:Citric_acid_cycle.
- Pyruvate_dehydrogenase_kinase wikiPageWikiLink Category:EC_2.7.11.
- Pyruvate_dehydrogenase_kinase wikiPageWikiLink Category:Glycolysis.
- Pyruvate_dehydrogenase_kinase wikiPageWikiLink Charcot–Marie–Tooth_disease.
- Pyruvate_dehydrogenase_kinase wikiPageWikiLink Citric_acid_cycle.
- Pyruvate_dehydrogenase_kinase wikiPageWikiLink Coenzyme_A.
- Pyruvate_dehydrogenase_kinase wikiPageWikiLink Cytosol.
- Pyruvate_dehydrogenase_kinase wikiPageWikiLink Diabetes_mellitus_type_2.
- Pyruvate_dehydrogenase_kinase wikiPageWikiLink Dichloroacetic_acid.
- Pyruvate_dehydrogenase_kinase wikiPageWikiLink Enzyme.
- Pyruvate_dehydrogenase_kinase wikiPageWikiLink Eukaryote.
- Pyruvate_dehydrogenase_kinase wikiPageWikiLink Glycolysis.
- Pyruvate_dehydrogenase_kinase wikiPageWikiLink Heart.
- Pyruvate_dehydrogenase_kinase wikiPageWikiLink Hydrogen_bond.
- Pyruvate_dehydrogenase_kinase wikiPageWikiLink Hyperglycemia.
- Pyruvate_dehydrogenase_kinase wikiPageWikiLink Hypoxia-inducible_factors.
- Pyruvate_dehydrogenase_kinase wikiPageWikiLink Insulin.
- Pyruvate_dehydrogenase_kinase wikiPageWikiLink Isozyme.
- Pyruvate_dehydrogenase_kinase wikiPageWikiLink Kinase.
- Pyruvate_dehydrogenase_kinase wikiPageWikiLink Lactic_acid.
- Pyruvate_dehydrogenase_kinase wikiPageWikiLink Lung.
- Pyruvate_dehydrogenase_kinase wikiPageWikiLink Mitochondrial_matrix.
- Pyruvate_dehydrogenase_kinase wikiPageWikiLink N-terminus.
- Pyruvate_dehydrogenase_kinase wikiPageWikiLink Nicotinamide_adenine_dinucleotide.
- Pyruvate_dehydrogenase_kinase wikiPageWikiLink PDK2.
- Pyruvate_dehydrogenase_kinase wikiPageWikiLink PDK3.
- Pyruvate_dehydrogenase_kinase wikiPageWikiLink PDK4.
- Pyruvate_dehydrogenase_kinase wikiPageWikiLink Phosphoinositide-dependent_kinase-1.
- Pyruvate_dehydrogenase_kinase wikiPageWikiLink Phosphorylation.
- Pyruvate_dehydrogenase_kinase wikiPageWikiLink Protein_phosphatase.
- Pyruvate_dehydrogenase_kinase wikiPageWikiLink Pyruvate_dehydrogenase.
- Pyruvate_dehydrogenase_kinase wikiPageWikiLink Pyruvate_dehydrogenase_complex.
- Pyruvate_dehydrogenase_kinase wikiPageWikiLink Pyruvate_dehydrogenase_lipoamide_kinase_isozyme_1.
- Pyruvate_dehydrogenase_kinase wikiPageWikiLink Pyruvate_dehydrogenase_phosphatase.
- Pyruvate_dehydrogenase_kinase wikiPageWikiLink Pyruvic_acid.
- Pyruvate_dehydrogenase_kinase wikiPageWikiLink Radicicol.
- Pyruvate_dehydrogenase_kinase wikiPageWikiLink Serine.
- Pyruvate_dehydrogenase_kinase wikiPageWikiLink Skeletal_muscle.
- Pyruvate_dehydrogenase_kinase wikiPageWikiLink Spleen.
- Pyruvate_dehydrogenase_kinase wikiPageWikiLink Steric_effects.
- Pyruvate_dehydrogenase_kinase wikiPageWikiLink Testicle.
- Pyruvate_dehydrogenase_kinase wikiPageWikiLink Tumor_hypoxia.
- Pyruvate_dehydrogenase_kinase wikiPageWikiLink File:Pyruvate_dehydrogenase_kinase_isozyme_4_with_bound_ADP.png.
- Pyruvate_dehydrogenase_kinase wikiPageWikiLinkText "Pyruvate dehydrogenase kinase".
- Pyruvate_dehydrogenase_kinase wikiPageWikiLinkText "pyruvate dehydrogenase kinase".
- Pyruvate_dehydrogenase_kinase caption "The areas around the three phosphorylation sites are shown in red. Site 1 is in the bottom left corner, site 2 in the top right, and site 3 in the bottom right.".
- Pyruvate_dehydrogenase_kinase casNumber "2620256".
- Pyruvate_dehydrogenase_kinase ecNumber "2.7".
- Pyruvate_dehydrogenase_kinase iubmbEcNumber "2".
- Pyruvate_dehydrogenase_kinase name "Pyruvate dehydrogenase kinase".
- Pyruvate_dehydrogenase_kinase wikiPageUsesTemplate Template:Citric_acid_cycle_enzymes.
- Pyruvate_dehydrogenase_kinase wikiPageUsesTemplate Template:EC_number.
- Pyruvate_dehydrogenase_kinase wikiPageUsesTemplate Template:Enzyme.
- Pyruvate_dehydrogenase_kinase wikiPageUsesTemplate Template:Enzymes.
- Pyruvate_dehydrogenase_kinase wikiPageUsesTemplate Template:MeshName.
- Pyruvate_dehydrogenase_kinase wikiPageUsesTemplate Template:Portal_bar.
- Pyruvate_dehydrogenase_kinase wikiPageUsesTemplate Template:Reflist.
- Pyruvate_dehydrogenase_kinase wikiPageUsesTemplate threonine-specific_protein_kinases.
- Pyruvate_dehydrogenase_kinase subject Category:Citric_acid_cycle.
- Pyruvate_dehydrogenase_kinase subject Category:EC_2.7.11.
- Pyruvate_dehydrogenase_kinase subject Category:Glycolysis.
- Pyruvate_dehydrogenase_kinase hypernym Enzyme.
- Pyruvate_dehydrogenase_kinase type Biomolecule.
- Pyruvate_dehydrogenase_kinase type Enzyme.
- Pyruvate_dehydrogenase_kinase type Protein.
- Pyruvate_dehydrogenase_kinase type Page.
- Pyruvate_dehydrogenase_kinase type Pathway.
- Pyruvate_dehydrogenase_kinase type Thing.
- Pyruvate_dehydrogenase_kinase type Q206229.
- Pyruvate_dehydrogenase_kinase type Q8047.
- Pyruvate_dehydrogenase_kinase comment "Pyruvate dehydrogenase kinase (also pyruvate dehydrogenase complex kinase, PDC kinase, or PDK; EC 2.7.11.2) is a kinase enzyme which acts to inactivate the enzyme pyruvate dehydrogenase by phosphorylating it using ATP. PDK thus participates in the regulation of the pyruvate dehydrogenase complex of which pyruvate dehydrogenase is the first component. Both PDK and the pyruvate dehydrogenase complex are located in the mitochondrial matrix of eukaryotes.".
- Pyruvate_dehydrogenase_kinase label "Pyruvate dehydrogenase kinase".
- Pyruvate_dehydrogenase_kinase sameAs Q6321025.
- Pyruvate_dehydrogenase_kinase sameAs Piruvato_deshidrogenasa_kinasa.
- Pyruvate_dehydrogenase_kinase sameAs Pyruvaattidehydrogenaasikinaasi.
- Pyruvate_dehydrogenase_kinase sameAs Pyruvate_déshydrogénase_kinase.
- Pyruvate_dehydrogenase_kinase sameAs Piruvat_dehidrogenase_kinase.
- Pyruvate_dehydrogenase_kinase sameAs Piruvato_desidrogenase_quinase.
- Pyruvate_dehydrogenase_kinase sameAs m.028cfs2.
- Pyruvate_dehydrogenase_kinase sameAs (Piruvat_dehidrogenaza_(acetil-transfer))_kinaza.
- Pyruvate_dehydrogenase_kinase sameAs (Piruvat_dehidrogenaza_(acetil-transfer))_kinaza.
- Pyruvate_dehydrogenase_kinase sameAs Q6321025.
- Pyruvate_dehydrogenase_kinase wasDerivedFrom Pyruvate_dehydrogenase_kinase?oldid=705521765.
- Pyruvate_dehydrogenase_kinase depiction Pyruvate_dehydrogenase_phosphorylation_sites.png.
- Pyruvate_dehydrogenase_kinase isPrimaryTopicOf Pyruvate_dehydrogenase_kinase.
- Pyruvate_dehydrogenase_kinase name "Pyruvate dehydrogenase kinase".