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- Partial_agonist abstract "In pharmacology, partial agonists are drugs that bind to and activate a given receptor, but have only partial efficacy at the receptor relative to a full agonist. They may also be considered ligands which display both agonistic and antagonistic effects — when both a full agonist and partial agonist are present, the partial agonist actually acts as a competitive antagonist, competing with the full agonist for receptor occupancy and producing a net decrease in the receptor activation observed with the full agonist alone. Clinically, partial agonists can be used to activate receptors to give a desired submaximal response when inadequate amounts of the endogenous ligand are present, or they can reduce the overstimulation of receptors when excess amounts of the endogenous ligand are present.Some currently common drugs that have been classed as partial agonists at particular receptors include buspirone, aripiprazole, buprenorphine, and norclozapine. Examples of ligands activating peroxisome proliferator-activated receptor gamma as partial agonists are honokiol and falcarindiol.".
- Partial_agonist thumbnail Agonist_2.png?width=300.
- Partial_agonist wikiPageID "791710".
- Partial_agonist wikiPageLength "3650".
- Partial_agonist wikiPageOutDegree "22".
- Partial_agonist wikiPageRevisionID "697296322".
- Partial_agonist wikiPageWikiLink Agonist.
- Partial_agonist wikiPageWikiLink Aripiprazole.
- Partial_agonist wikiPageWikiLink Beta_blocker.
- Partial_agonist wikiPageWikiLink Buprenorphine.
- Partial_agonist wikiPageWikiLink Buspirone.
- Partial_agonist wikiPageWikiLink Category:Pharmacodynamics.
- Partial_agonist wikiPageWikiLink Competitive_antagonist.
- Partial_agonist wikiPageWikiLink Desmethylclozapine.
- Partial_agonist wikiPageWikiLink Falcarindiol.
- Partial_agonist wikiPageWikiLink Honokiol.
- Partial_agonist wikiPageWikiLink Intrinsic_activity.
- Partial_agonist wikiPageWikiLink Inverse_agonist.
- Partial_agonist wikiPageWikiLink Ligand.
- Partial_agonist wikiPageWikiLink Peroxisome_proliferator-activated_receptor_gamma.
- Partial_agonist wikiPageWikiLink Pharmacology.
- Partial_agonist wikiPageWikiLink Receptor_(biochemistry).
- Partial_agonist wikiPageWikiLink Receptor_antagonist.
- Partial_agonist wikiPageWikiLink Selective_receptor_modulator.
- Partial_agonist wikiPageWikiLink File:Agonist_2.png.
- Partial_agonist wikiPageWikiLinkText "Partial agonist".
- Partial_agonist wikiPageWikiLinkText "agonist-antagonist".
- Partial_agonist wikiPageWikiLinkText "partial agonism".
- Partial_agonist wikiPageWikiLinkText "partial agonist".
- Partial_agonist wikiPageWikiLinkText "partial agonists".
- Partial_agonist wikiPageWikiLinkText "partial".
- Partial_agonist wikiPageUsesTemplate Template:Pharmacology.
- Partial_agonist wikiPageUsesTemplate Template:Pharmacology-stub.
- Partial_agonist wikiPageUsesTemplate Template:Reflist.
- Partial_agonist subject Category:Pharmacodynamics.
- Partial_agonist hypernym Drugs.
- Partial_agonist type Drug.
- Partial_agonist type Redirect.
- Partial_agonist type Science.
- Partial_agonist comment "In pharmacology, partial agonists are drugs that bind to and activate a given receptor, but have only partial efficacy at the receptor relative to a full agonist.".
- Partial_agonist label "Partial agonist".
- Partial_agonist sameAs Q770260.
- Partial_agonist sameAs Agonista_parcial.
- Partial_agonist sameAs Partialagonist.
- Partial_agonist sameAs Agonista_parcial.
- Partial_agonist sameAs آگونیست_نسبی.
- Partial_agonist sameAs Agoniste_partiel.
- Partial_agonist sameAs Agonista_parcial.
- Partial_agonist sameAs m.04n7hsl.
- Partial_agonist sameAs Частичный_агонист.
- Partial_agonist sameAs Parcijalni_agonist.
- Partial_agonist sameAs Parcijalni_agonist.
- Partial_agonist sameAs Q770260.
- Partial_agonist sameAs 部分激动剂.
- Partial_agonist wasDerivedFrom Partial_agonist?oldid=697296322.
- Partial_agonist depiction Agonist_2.png.
- Partial_agonist isPrimaryTopicOf Partial_agonist.