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- Norepinephrine–dopamine_disinhibitor abstract "Norepinephrine and dopamine disinhibitors (NDDIs) are a class of drugs which act at specific sites to disinhibit downstream norepinephrine and dopamine release in the brain.Agomelatine, an antidepressant which disinhibits norepinephrine and dopamine release in the frontal cortex by antagonizing 5-HT2C receptors, was the first drug to be described as an NDDI. While many other drugs also antagonize 5-HT2C receptors to some degree or another, they tend to be very non-specific in their actions, and as a result, the term \"NDDI\" has generally, though not always (for instance, fluoxetine has been called an NDDI in addition to SSRI due to its (weak) blockade of 5-HT2C), been reserved for describing newer, more selective agents in which disinhibition of norepinephrine and dopamine release is their primary mechanism of action.Another drug that has been referred to as an NDDI in the medical literature is flibanserin, which is approved as a treatment for hypoactive sexual desire disorder in premenopausal women. Flibanserin disinhibits norepinephrine and dopamine release in the prefrontal cortex by activating 5-HT1A receptors in this area.Aside from agomelatine, fluoxetine, and flibanserin, as of present, no other drugs have been described as NDDIs in the medical literature, despite the fact that many other existing drugs possess effects consistent with those of the definition of an NDDI. In any case, more drugs labeled specifically as NDDIs may be seen in the future.".
- Norepinephrine–dopamine_disinhibitor thumbnail Agomelatine.svg?width=300.
- Norepinephrine–dopamine_disinhibitor wikiPageID "25760657".
- Norepinephrine–dopamine_disinhibitor wikiPageLength "5344".
- Norepinephrine–dopamine_disinhibitor wikiPageOutDegree "27".
- Norepinephrine–dopamine_disinhibitor wikiPageRevisionID "678986101".
- Norepinephrine–dopamine_disinhibitor wikiPageWikiLink 5-HT1A_receptor.
- Norepinephrine–dopamine_disinhibitor wikiPageWikiLink 5-HT2C_receptor.
- Norepinephrine–dopamine_disinhibitor wikiPageWikiLink Agomelatine.
- Norepinephrine–dopamine_disinhibitor wikiPageWikiLink Antidepressant.
- Norepinephrine–dopamine_disinhibitor wikiPageWikiLink Binding_selectivity.
- Norepinephrine–dopamine_disinhibitor wikiPageWikiLink Brain.
- Norepinephrine–dopamine_disinhibitor wikiPageWikiLink Category:5-HT1A_agonists.
- Norepinephrine–dopamine_disinhibitor wikiPageWikiLink Category:5-HT2A_antagonists.
- Norepinephrine–dopamine_disinhibitor wikiPageWikiLink Category:5-HT2C_antagonists.
- Norepinephrine–dopamine_disinhibitor wikiPageWikiLink Category:Antidepressants.
- Norepinephrine–dopamine_disinhibitor wikiPageWikiLink Category:Female_sexual_dysfunction_drugs.
- Norepinephrine–dopamine_disinhibitor wikiPageWikiLink Dopamine.
- Norepinephrine–dopamine_disinhibitor wikiPageWikiLink Drug.
- Norepinephrine–dopamine_disinhibitor wikiPageWikiLink Flibanserin.
- Norepinephrine–dopamine_disinhibitor wikiPageWikiLink Fluoxetine.
- Norepinephrine–dopamine_disinhibitor wikiPageWikiLink Frontal_lobe.
- Norepinephrine–dopamine_disinhibitor wikiPageWikiLink Hypoactive_sexual_desire_disorder.
- Norepinephrine–dopamine_disinhibitor wikiPageWikiLink Mechanism_of_action.
- Norepinephrine–dopamine_disinhibitor wikiPageWikiLink Medical_literature.
- Norepinephrine–dopamine_disinhibitor wikiPageWikiLink Noradrenergic_and_specific_serotonergic_antidepressant.
- Norepinephrine–dopamine_disinhibitor wikiPageWikiLink Norepinephrine.
- Norepinephrine–dopamine_disinhibitor wikiPageWikiLink Prefrontal_cortex.
- Norepinephrine–dopamine_disinhibitor wikiPageWikiLink Receptor_antagonist.
- Norepinephrine–dopamine_disinhibitor wikiPageWikiLink Selective_serotonin_reuptake_inhibitor.
- Norepinephrine–dopamine_disinhibitor wikiPageWikiLink Serotonin_antagonist_and_reuptake_inhibitor.
- Norepinephrine–dopamine_disinhibitor wikiPageWikiLink Serotonin_modulator_and_stimulator.
- Norepinephrine–dopamine_disinhibitor wikiPageWikiLink File:Agomelatine.svg.
- Norepinephrine–dopamine_disinhibitor wikiPageWikiLinkText "Norepinephrine–dopamine disinhibitor".
- Norepinephrine–dopamine_disinhibitor wikiPageWikiLinkText "norepinephrine–dopamine disinhibitor".
- Norepinephrine–dopamine_disinhibitor wikiPageUsesTemplate Template:Antidepressants.
- Norepinephrine–dopamine_disinhibitor wikiPageUsesTemplate Template:Aphrodisiacs.
- Norepinephrine–dopamine_disinhibitor wikiPageUsesTemplate Template:Reflist.
- Norepinephrine–dopamine_disinhibitor wikiPageUsesTemplate Template:Serotonergics.
- Norepinephrine–dopamine_disinhibitor subject Category:5-HT1A_agonists.
- Norepinephrine–dopamine_disinhibitor subject Category:5-HT2A_antagonists.
- Norepinephrine–dopamine_disinhibitor subject Category:5-HT2C_antagonists.
- Norepinephrine–dopamine_disinhibitor subject Category:Antidepressants.
- Norepinephrine–dopamine_disinhibitor subject Category:Female_sexual_dysfunction_drugs.
- Norepinephrine–dopamine_disinhibitor hypernym Drugs.
- Norepinephrine–dopamine_disinhibitor type Drug.
- Norepinephrine–dopamine_disinhibitor type Agonist.
- Norepinephrine–dopamine_disinhibitor type Antagonist.
- Norepinephrine–dopamine_disinhibitor type Antidepressant.
- Norepinephrine–dopamine_disinhibitor type Drug.
- Norepinephrine–dopamine_disinhibitor type Psychoanaleptic.
- Norepinephrine–dopamine_disinhibitor comment "Norepinephrine and dopamine disinhibitors (NDDIs) are a class of drugs which act at specific sites to disinhibit downstream norepinephrine and dopamine release in the brain.Agomelatine, an antidepressant which disinhibits norepinephrine and dopamine release in the frontal cortex by antagonizing 5-HT2C receptors, was the first drug to be described as an NDDI.".
- Norepinephrine–dopamine_disinhibitor label "Norepinephrine–dopamine disinhibitor".
- Norepinephrine–dopamine_disinhibitor sameAs Q7050950.
- Norepinephrine–dopamine_disinhibitor sameAs m.09v5db7.
- Norepinephrine–dopamine_disinhibitor sameAs Q7050950.
- Norepinephrine–dopamine_disinhibitor wasDerivedFrom Norepinephrine–dopamine_disinhibitor?oldid=678986101.
- Norepinephrine–dopamine_disinhibitor depiction Agomelatine.svg.
- Norepinephrine–dopamine_disinhibitor isPrimaryTopicOf Norepinephrine–dopamine_disinhibitor.