Matches in DBpedia 2016-04 for { <http://dbpedia.org/resource/Fragment-based_lead_discovery> ?p ?o }
Showing triples 1 to 42 of
42
with 100 triples per page.
- Fragment-based_lead_discovery abstract "Fragment-based lead discovery (FBLD) also known as fragment-based drug discovery (FBDD) is a method used for finding lead compounds as part of the drug discovery process. It is based on identifying small chemical fragments, which may bind only weakly to the biological target, and then growing them or combining them to produce a lead with a higher affinity. FBLD can be compared with high-throughput screening (HTS). In HTS, libraries with up to millions of compounds, with molecular weights of around 500 Da, are screened, and nanomolar binding affinities are sought. In contrast, in the early phase of FBLD, libraries with a few thousand compounds with molecular weights of around 200 Da may be screened, and millimolar affinities can be considered useful.".
- Fragment-based_lead_discovery wikiPageID "18526787".
- Fragment-based_lead_discovery wikiPageLength "4559".
- Fragment-based_lead_discovery wikiPageOutDegree "17".
- Fragment-based_lead_discovery wikiPageRevisionID "594152607".
- Fragment-based_lead_discovery wikiPageWikiLink Atomic_mass_unit.
- Fragment-based_lead_discovery wikiPageWikiLink Biological_target.
- Fragment-based_lead_discovery wikiPageWikiLink Category:Biotechnology.
- Fragment-based_lead_discovery wikiPageWikiLink Category:Drug_discovery.
- Fragment-based_lead_discovery wikiPageWikiLink Drug_discovery.
- Fragment-based_lead_discovery wikiPageWikiLink Druglikeness.
- Fragment-based_lead_discovery wikiPageWikiLink Dynamic_combinatorial_chemistry.
- Fragment-based_lead_discovery wikiPageWikiLink Enthalpy.
- Fragment-based_lead_discovery wikiPageWikiLink Entropy.
- Fragment-based_lead_discovery wikiPageWikiLink High-throughput_screening.
- Fragment-based_lead_discovery wikiPageWikiLink Hydrogen_bond.
- Fragment-based_lead_discovery wikiPageWikiLink Lead_compound.
- Fragment-based_lead_discovery wikiPageWikiLink Ligand_efficiency.
- Fragment-based_lead_discovery wikiPageWikiLink Lipinskis_rule_of_five.
- Fragment-based_lead_discovery wikiPageWikiLink Molecular_mass.
- Fragment-based_lead_discovery wikiPageWikiLink Partition_coefficient.
- Fragment-based_lead_discovery wikiPageWikiLinkText "FBDD".
- Fragment-based_lead_discovery wikiPageWikiLinkText "Fragment-based lead discovery".
- Fragment-based_lead_discovery wikiPageWikiLinkText "fragment-based design".
- Fragment-based_lead_discovery wikiPageWikiLinkText "fragment-based lead discovery".
- Fragment-based_lead_discovery wikiPageWikiLinkText "fragments".
- Fragment-based_lead_discovery wikiPageUsesTemplate Template:Cite_book.
- Fragment-based_lead_discovery wikiPageUsesTemplate Template:Cite_journal.
- Fragment-based_lead_discovery wikiPageUsesTemplate Template:Refbegin.
- Fragment-based_lead_discovery wikiPageUsesTemplate Template:Refend.
- Fragment-based_lead_discovery wikiPageUsesTemplate Template:Reflist.
- Fragment-based_lead_discovery subject Category:Biotechnology.
- Fragment-based_lead_discovery subject Category:Drug_discovery.
- Fragment-based_lead_discovery hypernym Method.
- Fragment-based_lead_discovery type Software.
- Fragment-based_lead_discovery comment "Fragment-based lead discovery (FBLD) also known as fragment-based drug discovery (FBDD) is a method used for finding lead compounds as part of the drug discovery process. It is based on identifying small chemical fragments, which may bind only weakly to the biological target, and then growing them or combining them to produce a lead with a higher affinity. FBLD can be compared with high-throughput screening (HTS).".
- Fragment-based_lead_discovery label "Fragment-based lead discovery".
- Fragment-based_lead_discovery sameAs Q8565284.
- Fragment-based_lead_discovery sameAs m.04f5gb1.
- Fragment-based_lead_discovery sameAs Q8565284.
- Fragment-based_lead_discovery wasDerivedFrom Fragment-based_lead_discovery?oldid=594152607.
- Fragment-based_lead_discovery isPrimaryTopicOf Fragment-based_lead_discovery.