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- Discovery_and_development_of_phosphodiesterase_5_inhibitors abstract "Phosphodiesterases (PDEs) are a superfamily of enzymes. This superfamily is further classified into 11 families, PDE1 - PDE11, on the basis of regulatory properties, amino acid sequences, substrate specificities, pharmacological properties and tissue distribution. Their function is to degrade intracellular second messengers such as cyclic adenine monophosphate (cAMP) and cyclic guanosine monophosphate (cGMP) which leads to several biological processes like effect on intracellular calcium level by the Ca2+ pathway.Phosphodiesterase 5 (PDE5) is widely expressed in several tissues in the body for example brain, lung, kidney, urinary bladder, smooth muscle and platelets. It is possible to prevent cGMP hydrolysis by inhibiting PDE5 and therefore treat diseases associated with low cGMP levels, because of this, PDE5 is an ideal target for the development of inhibitors.The three major PDE5 inhibitors are sildenafil, tadalafil and vardenafil.".
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageExternalLink File:3D.Sild.2.png.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageExternalLink File:Figure_3._PDE5_Domains.png.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageExternalLink File:PDE5_SAR2.2.png.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageExternalLink Figure_5._PDE5_SAR1.png.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageID "41069188".
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageLength "21305".
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageOutDegree "63".
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageRevisionID "705165194".
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink African_trypanosomiasis.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink Alzheimers_disease.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink Amino_acid.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink CGMP-dependent_protein_kinase.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink CGMP-specific_phosphodiesterase_type_5.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink Category:Drug_discovery.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink Category:PDE5_inhibitors.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink Clinical_trial.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink Coronary_artery_disease.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink Cyclic_adenosine_monophosphate.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink Cyclic_guanosine_monophosphate.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink Endothelium.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink Enzyme.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink Erectile_dysfunction.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink Erection.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink Food_and_Drug_Administration.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink Guanylyl_cyclase.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink Hemodynamics.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink Hypotension.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink Methyl_group.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink Molecular_mass.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink Monomer.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink Negative_feedback.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink Neurotransmitter.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink Nitrate.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink Nitric_oxide.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink Oral_administration.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink PDE5_inhibitor.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink Parasitic_disease.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink Pfizer.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink Phosphodiesterase.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink Plasmodium_falciparum.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink Protein_dimer.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink Protein_superfamily.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink Prototype.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink Pulmonary_hypertension.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink Purine.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink Second_messenger_system.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink Serine.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink Sildenafil.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink Smooth_muscle_tissue.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink Structure–activity_relationship.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink Sulfonamide.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink Tadalafil.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink Vardenafil.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink File:3D.Sild.2.png.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink File:Biological_pathway_of_penile_erection.png.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink File:Figure_3._PDE5_Domains.png.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink File:Figure_5._PDE5_SAR1.png.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink File:PDE5_SAR2.2.png.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink File:PDE5_SAR3.png.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLink File:PDE5domains.png.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageWikiLinkText "PDE5 inhibitors".
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageUsesTemplate Template:Drug_design.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageUsesTemplate Template:Phosphodiesterase_inhibitors.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wikiPageUsesTemplate Template:Reflist.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors subject Category:Drug_discovery.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors subject Category:PDE5_inhibitors.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors comment "Phosphodiesterases (PDEs) are a superfamily of enzymes. This superfamily is further classified into 11 families, PDE1 - PDE11, on the basis of regulatory properties, amino acid sequences, substrate specificities, pharmacological properties and tissue distribution.".
- Discovery_and_development_of_phosphodiesterase_5_inhibitors label "Discovery and development of phosphodiesterase 5 inhibitors".
- Discovery_and_development_of_phosphodiesterase_5_inhibitors sameAs Q16154408.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors sameAs m.0z6sgq6.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors sameAs Q16154408.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors wasDerivedFrom Discovery_and_development_of_phosphodiesterase_5_inhibitors?oldid=705165194.
- Discovery_and_development_of_phosphodiesterase_5_inhibitors isPrimaryTopicOf Discovery_and_development_of_phosphodiesterase_5_inhibitors.