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- Discovery_and_development_of_memantine_and_related_compounds abstract "In 1972 a possible therapeutic importance of memantine, an adamantane derivative, was discovered for treating neurodegenerative disorders. Since 1989 memantine has been recognized to be an uncompetitive antagonist of the N-methyl-D-aspartate receptor (NMDA receptor), entering the channel of the receptor after it’s been activated and thereby blocking the flow of ions.The NMDA receptor channels play an important role in synaptic plasticity and synapse formation underlying memory, learning and formation of neural networks during development in the central nervous system (CNS). Overactivation of the receptor, causing excessive influx of Ca2+ can lead to excitotoxicity which is implied to be involved in some neurodegenerative disorders. Blocking of NMDA receptors could therefore, in theory, be useful in treating such diseases.The main problem with the development of NMDA receptor antagonist for neuroprotection is that the physiological NMDA receptor activity is essential for normal neuronal function. To be clinically accepted the antagonists must block excessive activation without blocking the normal function.".
- Discovery_and_development_of_memantine_and_related_compounds thumbnail NR1-NR2B_subunit.jpg?width=300.
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- Discovery_and_development_of_memantine_and_related_compounds wikiPageLength "25074".
- Discovery_and_development_of_memantine_and_related_compounds wikiPageOutDegree "65".
- Discovery_and_development_of_memantine_and_related_compounds wikiPageRevisionID "691521319".
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink AMPA_receptor.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink Adamantane.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink Agonist.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink Alzheimers_disease.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink Amantadine.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink Amyotrophic_lateral_sclerosis.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink Anesthesia.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink Anesthetic.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink Antagonist.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink Anticholinergic.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink Binding_site.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink Category:Drug_discovery.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink Central_nervous_system.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink Clinical_trial.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink Competitiveness.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink Cyclohexane.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink Depolarization.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink Dizocilpine.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink Dopaminergic.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink Efficacy.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink Epilepsy.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink Excitotoxicity.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink GRIN2B.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink Glutamic_acid.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink Glycine.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink Hallucination.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink Huntingtons_disease.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink Hypoglycemia.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink Hypotension.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink IC50.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink In_vitro.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink In_vivo.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink Ion_channel.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink Ketamine.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink Medicinal_chemistry.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink Memantine.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink NMDA_receptor.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink NMDA_receptor_antagonist.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink Neramexane.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink Neurodegeneration.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink Neurological_disorder.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink Neuroprotection.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink Neurotoxicity.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink Nitromemantine.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink Nitrosylation.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink Parkinsons_disease.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink Patch_clamp.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink Phencyclidine.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink Serine.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink Structure–activity_relationship.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink Synaptic_plasticity.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink Uncompetitive_antagonist.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink File:Memantine_and_amantadine.jpg.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink File:NMDA_receptor_antagonist.jpg.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink File:NR1-NR2B_subunit.jpg.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink File:NR1-NR2B_subunit.png.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink File:Neramexane.jpg.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink File:Nitromemantine.jpg.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageWikiLink File:SAR_of_amantadine_and_related_compunds.jpg.
- Discovery_and_development_of_memantine_and_related_compounds wikiPageUsesTemplate Template:Reflist.
- Discovery_and_development_of_memantine_and_related_compounds subject Category:Drug_discovery.
- Discovery_and_development_of_memantine_and_related_compounds comment "In 1972 a possible therapeutic importance of memantine, an adamantane derivative, was discovered for treating neurodegenerative disorders.".
- Discovery_and_development_of_memantine_and_related_compounds label "Discovery and development of memantine and related compounds".
- Discovery_and_development_of_memantine_and_related_compounds wasDerivedFrom Discovery_and_development_of_memantine_and_related_compounds?oldid=691521319.
- Discovery_and_development_of_memantine_and_related_compounds depiction NR1-NR2B_subunit.jpg.
- Discovery_and_development_of_memantine_and_related_compounds isPrimaryTopicOf Discovery_and_development_of_memantine_and_related_compounds.