Matches in DBpedia 2016-04 for { <http://dbpedia.org/resource/CYP2D6> ?p ?o }
- CYP2D6 abstract "Cytochrome P450 2D6 is an enzyme that in humans is encoded by the CYP2D6 gene. CYP2D6 is primarily expressed in the liver. It is also highly expressed in areas of the CNS, including the substantia nigra.CYP2D6, a member of the cytochrome P450 mixed-function oxidase system, is one of the most important enzymes involved in the metabolism of xenobiotics in the body. In particular, CYP2D6 is responsible for the metabolism and elimination of approximately 25% of clinically used drugs, in a process referred to as O-demethylation. This enzyme also metabolizes several endogenous substances such as hydroxytryptamines and neurosteroids.There is considerable variation in the efficiency and amount of CYP2D6 enzyme produced between individuals. Hence for drugs that are metabolized by CYP2D6 (that is, are CYP2D6 substrates), certain individuals will eliminate these drugs quickly (ultrarapid metabolizers) while others slowly (poor metabolizers). If a drug is metabolized too quickly, it may decrease the drug's efficacy while if the drug is metabolized too slowly, toxicity may result. Hence the dose of the drug may have to be adjusted to take into account of the speed at which it is metabolized by CYP2D6.In addition, other drugs may function as inhibitors of CYP2D6 activity or inducers of CYP2D6 enzyme expression that will lead to decreased or increased CYP2D6 activity respectively. If such a drug is taken at the same time a second drug that is a CYP2D6 substrate, the first drug may affect the elimination rate of the second through what is known as a drug-drug interaction.".
- CYP2D6 entrezgene "1565".
- CYP2D6 wikiPageExternalLink 2D6sub.
- CYP2D6 wikiPageExternalLink index.jsp.
- CYP2D6 wikiPageID "1024815".
- CYP2D6 wikiPageLength "26170".
- CYP2D6 wikiPageOutDegree "213".
- CYP2D6 wikiPageRevisionID "703466109".
- CYP2D6 wikiPageWikiLink 5-HT3_antagonist.
- CYP2D6 wikiPageWikiLink Acetylcholinesterase_inhibitor.
- CYP2D6 wikiPageWikiLink Activation.
- CYP2D6 wikiPageWikiLink Addiction.
- CYP2D6 wikiPageWikiLink African_Americans.
- CYP2D6 wikiPageWikiLink Allele.
- CYP2D6 wikiPageWikiLink Alpha-adrenergic_agonist.
- CYP2D6 wikiPageWikiLink Alprenolol.
- CYP2D6 wikiPageWikiLink Alternative_splicing.
- CYP2D6 wikiPageWikiLink Amiodarone.
- CYP2D6 wikiPageWikiLink Amitriptyline.
- CYP2D6 wikiPageWikiLink Amphetamine.
- CYP2D6 wikiPageWikiLink Analgesic.
- CYP2D6 wikiPageWikiLink Anorectic.
- CYP2D6 wikiPageWikiLink Anti-diabetic_medication.
- CYP2D6 wikiPageWikiLink Antianginal.
- CYP2D6 wikiPageWikiLink Antiarrhythmic_agent.
- CYP2D6 wikiPageWikiLink Anticholinergic.
- CYP2D6 wikiPageWikiLink Antidepressant.
- CYP2D6 wikiPageWikiLink Antiemetic.
- CYP2D6 wikiPageWikiLink Antifungal.
- CYP2D6 wikiPageWikiLink Antihistamine.
- CYP2D6 wikiPageWikiLink Antihypertensive_drug.
- CYP2D6 wikiPageWikiLink Antiplatelet_drug.
- CYP2D6 wikiPageWikiLink Antipsychotic.
- CYP2D6 wikiPageWikiLink Anxiolytic.
- CYP2D6 wikiPageWikiLink Area_under_the_curve_(pharmacokinetics).
- CYP2D6 wikiPageWikiLink Aripiprazole.
- CYP2D6 wikiPageWikiLink Asian_people.
- CYP2D6 wikiPageWikiLink Atomoxetine.
- CYP2D6 wikiPageWikiLink Bactericide.
- CYP2D6 wikiPageWikiLink Beta_blocker.
- CYP2D6 wikiPageWikiLink Bufuralol.
- CYP2D6 wikiPageWikiLink Buprenorphine.
- CYP2D6 wikiPageWikiLink Bupropion.
- CYP2D6 wikiPageWikiLink Calcium_channel_blocker.
- CYP2D6 wikiPageWikiLink Cannabidiol.
- CYP2D6 wikiPageWikiLink Cannabinoid.
- CYP2D6 wikiPageWikiLink Carvedilol.
- CYP2D6 wikiPageWikiLink Category:Amphetamine.
- CYP2D6 wikiPageWikiLink Category:Cytochrome_P450.
- CYP2D6 wikiPageWikiLink Category:EC_1.14.14.
- CYP2D6 wikiPageWikiLink Celecoxib.
- CYP2D6 wikiPageWikiLink Chemotherapy.
- CYP2D6 wikiPageWikiLink Chlorphenamine.
- CYP2D6 wikiPageWikiLink Chlorpromazine.
- CYP2D6 wikiPageWikiLink Chromosome_22_(human).
- CYP2D6 wikiPageWikiLink Cimetidine.
- CYP2D6 wikiPageWikiLink Cinacalcet.
- CYP2D6 wikiPageWikiLink Citalopram.
- CYP2D6 wikiPageWikiLink Clearance_(medicine).
- CYP2D6 wikiPageWikiLink Clemastine.
- CYP2D6 wikiPageWikiLink Clomipramine.
- CYP2D6 wikiPageWikiLink Cocaine.
- CYP2D6 wikiPageWikiLink Codeine.
- CYP2D6 wikiPageWikiLink Cough_medicine.
- CYP2D6 wikiPageWikiLink Cytochrome_P450.
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- CYP2D6 wikiPageWikiLink Dextromethorphan.
- CYP2D6 wikiPageWikiLink Diphenhydramine.
- CYP2D6 wikiPageWikiLink Donepezil.
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- CYP2D6 wikiPageWikiLink Doxorubicin.
- CYP2D6 wikiPageWikiLink Drug_interaction.
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- CYP2D6 wikiPageWikiLink Enzyme.
- CYP2D6 wikiPageWikiLink Enzyme_induction_and_inhibition.
- CYP2D6 wikiPageWikiLink Enzyme_inhibitor.
- CYP2D6 wikiPageWikiLink Escitalopram.
- CYP2D6 wikiPageWikiLink Flecainide.
- CYP2D6 wikiPageWikiLink Fluoxetine.
- CYP2D6 wikiPageWikiLink Fluvoxamine.
- CYP2D6 wikiPageWikiLink Gene.
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- CYP2D6 wikiPageWikiLink Genotype.
- CYP2D6 wikiPageWikiLink Glucocorticoid.
- CYP2D6 wikiPageWikiLink Glutethimide.
- CYP2D6 wikiPageWikiLink H1_antagonist.
- CYP2D6 wikiPageWikiLink H2_antagonist.
- CYP2D6 wikiPageWikiLink Halofantrine.
- CYP2D6 wikiPageWikiLink Haloperidol.
- CYP2D6 wikiPageWikiLink Hydrocodone.
- CYP2D6 wikiPageWikiLink Hydroxyzine.
- CYP2D6 wikiPageWikiLink Hyperforin.
- CYP2D6 wikiPageWikiLink Hypericum_perforatum.
- CYP2D6 wikiPageWikiLink Hypnotic.
- CYP2D6 wikiPageWikiLink Iloperidone.