Matches in DBpedia 2016-04 for { <http://dbpedia.org/resource/C-Met_inhibitors> ?p ?o }
- C-Met_inhibitors abstract "c-Met inhibitors are a class of small molecules that inhibit the enzymatic activity of the c-Met tyrosine kinase. These inhibitors may have therapeutic application in the treatment of various types of cancers.Many c-Met inhibitors are currently in clinical trials. Cabozantinib was the first to be approved by the U.S. FDA; approved in November 2012 for the treatment of medullary thyroid cancer and it has also started clinical trials for the treatment of prostate, bladder, ovarian, brain, melanoma, breast, non-small cell lung, pancreatic, hepatocellular and kidney cancers.c-Met stimulates cell scattering, invasion, protection from apoptosis and angiogenesis. c-Met is a receptor tyrosine kinase, which can cause a wide variety of different cancers, such as renal, gastric and small cell lung carcinomas, central nervous system tumours, as well as several sarcomas when its activity is dysregulated. Targeting the ATP binding site of c-Met by small molecules inhibitors is one strategy for inhibition of the tyrosine kinase.".
- C-Met_inhibitors thumbnail K252_and_c-met.png?width=300.
- C-Met_inhibitors wikiPageExternalLink Home.
- C-Met_inhibitors wikiPageID "33238902".
- C-Met_inhibitors wikiPageLength "29866".
- C-Met_inhibitors wikiPageOutDegree "118".
- C-Met_inhibitors wikiPageRevisionID "706103613".
- C-Met_inhibitors wikiPageWikiLink 5-HT3_antagonist.
- C-Met_inhibitors wikiPageWikiLink AMG_458.
- C-Met_inhibitors wikiPageWikiLink Acyl.
- C-Met_inhibitors wikiPageWikiLink Adenosine_triphosphate.
- C-Met_inhibitors wikiPageWikiLink Agonist.
- C-Met_inhibitors wikiPageWikiLink Amine.
- C-Met_inhibitors wikiPageWikiLink Anaplastic_lymphoma_kinase.
- C-Met_inhibitors wikiPageWikiLink Angiogenesis.
- C-Met_inhibitors wikiPageWikiLink Antibody.
- C-Met_inhibitors wikiPageWikiLink Apoptosis.
- C-Met_inhibitors wikiPageWikiLink Aryl.
- C-Met_inhibitors wikiPageWikiLink Autophosphorylation.
- C-Met_inhibitors wikiPageWikiLink Benzyl.
- C-Met_inhibitors wikiPageWikiLink Bioavailability.
- C-Met_inhibitors wikiPageWikiLink C-Met.
- C-Met_inhibitors wikiPageWikiLink CCR5_receptor_antagonist.
- C-Met_inhibitors wikiPageWikiLink Cabozantinib.
- C-Met_inhibitors wikiPageWikiLink Cannabinoid_receptor_antagonist.
- C-Met_inhibitors wikiPageWikiLink Catalysis.
- C-Met_inhibitors wikiPageWikiLink Category:Cancer_research.
- C-Met_inhibitors wikiPageWikiLink Category:Protein_kinase_inhibitors.
- C-Met_inhibitors wikiPageWikiLink Cell_growth.
- C-Met_inhibitors wikiPageWikiLink Central_nervous_system.
- C-Met_inhibitors wikiPageWikiLink Chemotherapy.
- C-Met_inhibitors wikiPageWikiLink Clinical_trial.
- C-Met_inhibitors wikiPageWikiLink Competitive_inhibition.
- C-Met_inhibitors wikiPageWikiLink Cytoskeleton.
- C-Met_inhibitors wikiPageWikiLink Development_of_dipeptidyl_peptidase-4_inhibitors.
- C-Met_inhibitors wikiPageWikiLink Discovery_and_development_of_HIV-protease_inhibitors.
- C-Met_inhibitors wikiPageWikiLink Discovery_and_development_of_TRPV1_antagonists.
- C-Met_inhibitors wikiPageWikiLink Discovery_and_development_of_cyclooxygenase_2_inhibitors.
- C-Met_inhibitors wikiPageWikiLink Discovery_and_development_of_non-nucleoside_reverse-transcriptase_inhibitors.
- C-Met_inhibitors wikiPageWikiLink Embryo.
- C-Met_inhibitors wikiPageWikiLink Enzyme_inhibitor.
- C-Met_inhibitors wikiPageWikiLink Epithelial–mesenchymal_transition.
- C-Met_inhibitors wikiPageWikiLink Epithelium.
- C-Met_inhibitors wikiPageWikiLink Fibroblast.
- C-Met_inhibitors wikiPageWikiLink Fluorine.
- C-Met_inhibitors wikiPageWikiLink Food_and_Drug_Administration.
- C-Met_inhibitors wikiPageWikiLink Foretinib.
- C-Met_inhibitors wikiPageWikiLink Half-life.
- C-Met_inhibitors wikiPageWikiLink Hepatocyte_growth_factor.
- C-Met_inhibitors wikiPageWikiLink Heterocyclic_compound.
- C-Met_inhibitors wikiPageWikiLink Hydrogen_bond.
- C-Met_inhibitors wikiPageWikiLink Hydrophobe.
- C-Met_inhibitors wikiPageWikiLink Immunotherapy.
- C-Met_inhibitors wikiPageWikiLink In_vivo.
- C-Met_inhibitors wikiPageWikiLink Intracellular.
- C-Met_inhibitors wikiPageWikiLink JNJ-38877605.
- C-Met_inhibitors wikiPageWikiLink K252a.
- C-Met_inhibitors wikiPageWikiLink Ligand.
- C-Met_inhibitors wikiPageWikiLink Liver.
- C-Met_inhibitors wikiPageWikiLink MK-2461.
- C-Met_inhibitors wikiPageWikiLink MTOR_inhibitors.
- C-Met_inhibitors wikiPageWikiLink Mammal.
- C-Met_inhibitors wikiPageWikiLink Medullary_thyroid_cancer.
- C-Met_inhibitors wikiPageWikiLink Melatonin_receptor_agonist.
- C-Met_inhibitors wikiPageWikiLink Mesenchymal_stem_cell.
- C-Met_inhibitors wikiPageWikiLink Mesenchymal–epithelial_transition.
- C-Met_inhibitors wikiPageWikiLink Metastasis.
- C-Met_inhibitors wikiPageWikiLink Molecule.
- C-Met_inhibitors wikiPageWikiLink Morphogenesis.
- C-Met_inhibitors wikiPageWikiLink Mutation.
- C-Met_inhibitors wikiPageWikiLink Non-competitive_inhibition.
- C-Met_inhibitors wikiPageWikiLink Non-small-cell_lung_carcinoma.
- C-Met_inhibitors wikiPageWikiLink Oncogene.
- C-Met_inhibitors wikiPageWikiLink PF-04217903.
- C-Met_inhibitors wikiPageWikiLink Pharmaceutical_industry.
- C-Met_inhibitors wikiPageWikiLink Pharmacokinetics.
- C-Met_inhibitors wikiPageWikiLink Phenol.
- C-Met_inhibitors wikiPageWikiLink Phosphorylation.
- C-Met_inhibitors wikiPageWikiLink Prognosis.
- C-Met_inhibitors wikiPageWikiLink Protein.
- C-Met_inhibitors wikiPageWikiLink Purine.
- C-Met_inhibitors wikiPageWikiLink Pyridine.
- C-Met_inhibitors wikiPageWikiLink Pyrimidone.
- C-Met_inhibitors wikiPageWikiLink Pyrrole.
- C-Met_inhibitors wikiPageWikiLink Quinoline.
- C-Met_inhibitors wikiPageWikiLink Radiation_therapy.
- C-Met_inhibitors wikiPageWikiLink Receptor_tyrosine_kinase.
- C-Met_inhibitors wikiPageWikiLink Renal_cell_carcinoma.
- C-Met_inhibitors wikiPageWikiLink Ribose.
- C-Met_inhibitors wikiPageWikiLink Sarcoma.
- C-Met_inhibitors wikiPageWikiLink Small-cell_carcinoma.
- C-Met_inhibitors wikiPageWikiLink Small_molecule.
- C-Met_inhibitors wikiPageWikiLink Staurosporine.
- C-Met_inhibitors wikiPageWikiLink Stomach_cancer.
- C-Met_inhibitors wikiPageWikiLink Structure–activity_relationship.
- C-Met_inhibitors wikiPageWikiLink Substrate_(chemistry).
- C-Met_inhibitors wikiPageWikiLink Sulfonamide.
- C-Met_inhibitors wikiPageWikiLink Thiourea.
- C-Met_inhibitors wikiPageWikiLink Tivantinib.
- C-Met_inhibitors wikiPageWikiLink Triazine.