Matches in DBpedia 2016-04 for { <http://dbpedia.org/resource/5-HT2c_receptor_agonist> ?p ?o }
- 5-HT2c_receptor_agonist abstract "Serotonin 5-HT2 receptors are stimulated by monoamine neurotransmitters including serotonin, dopamine and norepinephrine. 5-HT2 receptor stimulation causes a buildup of intracellular inositol triphosphate and thereby an increase of cytosolic Ca2+. 5-HT2C receptor agonists are attractive drug targets that have potential use in the treatment of a number of conditions including obesity, psychiatric disorders, sexual dysfunction and urinary incontinence.The 5-HT2C receptors are one of three subtypes that belong to the serotonin 5-HT2 receptor subfamily along with 5-HT2A and 5-HT2B receptors. The development of 5-HT2C agonists has been a major obstacle, because of severe side effects due to a lack of selectivity over 5-HT2A and 5-HT2B receptors. Activation of 5-HT2A receptors can induce hallucinations, and the activation of 5-HT2B receptors has been implicated in cardiac valvular insufficiency and possibly in pulmonary hypertension.".
- 5-HT2c_receptor_agonist wikiPageID "37051328".
- 5-HT2c_receptor_agonist wikiPageLength "46622".
- 5-HT2c_receptor_agonist wikiPageOutDegree "119".
- 5-HT2c_receptor_agonist wikiPageRevisionID "699787859".
- 5-HT2c_receptor_agonist wikiPageWikiLink 5-HT2A_receptor.
- 5-HT2c_receptor_agonist wikiPageWikiLink 5-HT2B_receptor.
- 5-HT2c_receptor_agonist wikiPageWikiLink 5-HT2C_receptor.
- 5-HT2c_receptor_agonist wikiPageWikiLink 5-HT2_receptor.
- 5-HT2c_receptor_agonist wikiPageWikiLink 5-HT_receptor.
- 5-HT2c_receptor_agonist wikiPageWikiLink Agonist.
- 5-HT2c_receptor_agonist wikiPageWikiLink Aliphatic_compound.
- 5-HT2c_receptor_agonist wikiPageWikiLink Amygdala.
- 5-HT2c_receptor_agonist wikiPageWikiLink Animal_locomotion.
- 5-HT2c_receptor_agonist wikiPageWikiLink Anorectic.
- 5-HT2c_receptor_agonist wikiPageWikiLink Antagonist.
- 5-HT2c_receptor_agonist wikiPageWikiLink Anti-obesity_medication.
- 5-HT2c_receptor_agonist wikiPageWikiLink Antipsychotic.
- 5-HT2c_receptor_agonist wikiPageWikiLink Atypical_antipsychotic.
- 5-HT2c_receptor_agonist wikiPageWikiLink Behavioural_despair_test.
- 5-HT2c_receptor_agonist wikiPageWikiLink Benzofuran.
- 5-HT2c_receptor_agonist wikiPageWikiLink Binding_constant.
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- 5-HT2c_receptor_agonist wikiPageWikiLink Category:5-HT2C_agonists.
- 5-HT2c_receptor_agonist wikiPageWikiLink Category:Antiobesity_drugs.
- 5-HT2c_receptor_agonist wikiPageWikiLink Category:Drug_discovery.
- 5-HT2c_receptor_agonist wikiPageWikiLink Category:Receptor_agonists.
- 5-HT2c_receptor_agonist wikiPageWikiLink Chemical_compound.
- 5-HT2c_receptor_agonist wikiPageWikiLink Chemical_synapse.
- 5-HT2c_receptor_agonist wikiPageWikiLink Choroid_plexus.
- 5-HT2c_receptor_agonist wikiPageWikiLink Clinical_trial.
- 5-HT2c_receptor_agonist wikiPageWikiLink Cytosol.
- 5-HT2c_receptor_agonist wikiPageWikiLink Dexfenfluramine.
- 5-HT2c_receptor_agonist wikiPageWikiLink Diazepine.
- 5-HT2c_receptor_agonist wikiPageWikiLink Dopamine.
- 5-HT2c_receptor_agonist wikiPageWikiLink Dorsomedial_hypothalamic_nucleus.
- 5-HT2c_receptor_agonist wikiPageWikiLink Enantiomer.
- 5-HT2c_receptor_agonist wikiPageWikiLink Endogeny_(biology).
- 5-HT2c_receptor_agonist wikiPageWikiLink Energy_homeostasis.
- 5-HT2c_receptor_agonist wikiPageWikiLink Exogeny.
- 5-HT2c_receptor_agonist wikiPageWikiLink Extracellular_signal-regulated_kinases.
- 5-HT2c_receptor_agonist wikiPageWikiLink Fenfluramine.
- 5-HT2c_receptor_agonist wikiPageWikiLink phentermine.
- 5-HT2c_receptor_agonist wikiPageWikiLink Food_and_Drug_Administration.
- 5-HT2c_receptor_agonist wikiPageWikiLink G_protein–coupled_receptor.
- 5-HT2c_receptor_agonist wikiPageWikiLink Gq_alpha_subunit.
- 5-HT2c_receptor_agonist wikiPageWikiLink Homology_(biology).
- 5-HT2c_receptor_agonist wikiPageWikiLink Hydrogen_bond.
- 5-HT2c_receptor_agonist wikiPageWikiLink Hypoactivity.
- 5-HT2c_receptor_agonist wikiPageWikiLink Indole.
- 5-HT2c_receptor_agonist wikiPageWikiLink Inositol_trisphosphate.
- 5-HT2c_receptor_agonist wikiPageWikiLink Inverse_agonist.
- 5-HT2c_receptor_agonist wikiPageWikiLink Knockout_mouse.
- 5-HT2c_receptor_agonist wikiPageWikiLink Leptin.
- 5-HT2c_receptor_agonist wikiPageWikiLink Levofenfluramine.
- 5-HT2c_receptor_agonist wikiPageWikiLink Ligand.
- 5-HT2c_receptor_agonist wikiPageWikiLink Lorcaserin.
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- 5-HT2c_receptor_agonist wikiPageWikiLink Mesolimbic_pathway.
- 5-HT2c_receptor_agonist wikiPageWikiLink Meta-Chlorophenylpiperazine.
- 5-HT2c_receptor_agonist wikiPageWikiLink Monoamine_neurotransmitter.
- 5-HT2c_receptor_agonist wikiPageWikiLink Mood_stabilizer.
- 5-HT2c_receptor_agonist wikiPageWikiLink Neuroplasticity.
- 5-HT2c_receptor_agonist wikiPageWikiLink Neurotrophin.
- 5-HT2c_receptor_agonist wikiPageWikiLink Nigrostriatal_pathway.
- 5-HT2c_receptor_agonist wikiPageWikiLink Norepinephrine.
- 5-HT2c_receptor_agonist wikiPageWikiLink Obesity.
- 5-HT2c_receptor_agonist wikiPageWikiLink PRX-00933.
- 5-HT2c_receptor_agonist wikiPageWikiLink Paraventricular_nucleus_of_hypothalamus.
- 5-HT2c_receptor_agonist wikiPageWikiLink Partial_agonist.
- 5-HT2c_receptor_agonist wikiPageWikiLink Pharmacophore.
- 5-HT2c_receptor_agonist wikiPageWikiLink Phentermine.
- 5-HT2c_receptor_agonist wikiPageWikiLink Phenylalanine.
- 5-HT2c_receptor_agonist wikiPageWikiLink Phosphatidylinositol_4,5-bisphosphate.
- 5-HT2c_receptor_agonist wikiPageWikiLink Phospholipase_A2.
- 5-HT2c_receptor_agonist wikiPageWikiLink Phospholipase_C.
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- 5-HT2c_receptor_agonist wikiPageWikiLink Piperazine.
- 5-HT2c_receptor_agonist wikiPageWikiLink Polyphagia.
- 5-HT2c_receptor_agonist wikiPageWikiLink Pre-clinical_development.
- 5-HT2c_receptor_agonist wikiPageWikiLink RHOA.
- 5-HT2c_receptor_agonist wikiPageWikiLink Racemic_mixture.
- 5-HT2c_receptor_agonist wikiPageWikiLink Redox.
- 5-HT2c_receptor_agonist wikiPageWikiLink Regeneration_(biology).
- 5-HT2c_receptor_agonist wikiPageWikiLink Reuptake.
- 5-HT2c_receptor_agonist wikiPageWikiLink Ro60-0175.
- 5-HT2c_receptor_agonist wikiPageWikiLink SB-242084.
- 5-HT2c_receptor_agonist wikiPageWikiLink SB-243213.
- 5-HT2c_receptor_agonist wikiPageWikiLink Salt_bridge.
- 5-HT2c_receptor_agonist wikiPageWikiLink Selective_serotonin_reuptake_inhibitor.
- 5-HT2c_receptor_agonist wikiPageWikiLink Serotonin.
- 5-HT2c_receptor_agonist wikiPageWikiLink Serotonin_antagonist.
- 5-HT2c_receptor_agonist wikiPageWikiLink Serotonin_receptor_agonist.
- 5-HT2c_receptor_agonist wikiPageWikiLink Sexual_dysfunction.
- 5-HT2c_receptor_agonist wikiPageWikiLink Solitary_tract.
- 5-HT2c_receptor_agonist wikiPageWikiLink Stress_incontinence.
- 5-HT2c_receptor_agonist wikiPageWikiLink Structure–activity_relationship.
- 5-HT2c_receptor_agonist wikiPageWikiLink Urinary_incontinence.
- 5-HT2c_receptor_agonist wikiPageWikiLink Urination.
- 5-HT2c_receptor_agonist wikiPageWikiLink Vabicaserin.