Matches in DBpedia 2015-10 for { <http://dbpedia.org/resource/Trace_amine> ?p ?o }
- Trace_amine abstract "Trace amines are an endogenous group of trace amine associated receptor 1 (TAAR1) agonists – and hence, monoaminergic neuromodulators – that are structurally and metabolically related to classical monoamine neurotransmitters. Compared to the classical monoamines, they are present in trace concentrations. They are distributed heterogeneously throughout the mammalian brain and peripheral nervous tissues and exhibit high rates of metabolism. Although they can be synthesized within parent monoamine neurotransmitter systems, there is evidence that suggests that some of them may comprise their own independent neurotransmitter systems.Trace amines play significant roles in regulating the quantity of neurotransmitters in the synaptic cleft of monoamine neurons with co-localized TAAR1. They have well-characterized presynaptic amphetamine-like effects on these monoamine neurons via TAAR1 activation; specifically, they release and prevent reuptake of neurotransmitters from the synaptic cleft. Phenethylamine even happens to have the same pharmacodynamics as regular amphetamine in human dopamine neurons, as both compounds induce efflux from vesicular monoamine transporter 2 (VMAT2) and activate TAAR1 with comparable efficacy. Like dopamine, noradrenaline, and serotonin, the trace amines have been implicated in a vast array of human disorders of affect and cognition, such as ADHD, depression and schizophrenia, among others. Trace aminergic hypo-function is particularly relevant to ADHD, since the two most commonly prescribed drugs for ADHD, amphetamine and methylphenidate, increase phenethylamine biosynthesis in treatment-responsive individuals with ADHD.A thorough review of trace amine-associated receptors that discusses the historical evolution of this research particularly well is that of Grandy.".
- Trace_amine thumbnail Phenethylamine2DCSD.svg?width=300.
- Trace_amine wikiPageID "5552077".
- Trace_amine wikiPageLength "14673".
- Trace_amine wikiPageOutDegree "54".
- Trace_amine wikiPageRevisionID "676343697".
- Trace_amine wikiPageWikiLink 3-Iodothyronamine.
- Trace_amine wikiPageWikiLink 3-Methoxytyramine.
- Trace_amine wikiPageWikiLink ADHD.
- Trace_amine wikiPageWikiLink Amphetamine.
- Trace_amine wikiPageWikiLink Attention_deficit_hyperactivity_disorder.
- Trace_amine wikiPageWikiLink Catecholamine.
- Trace_amine wikiPageWikiLink Category:Amines.
- Trace_amine wikiPageWikiLink Category:Amphetamine.
- Trace_amine wikiPageWikiLink Category:Neurochemistry.
- Trace_amine wikiPageWikiLink Category:Neurotransmitters.
- Trace_amine wikiPageWikiLink Category:TAAR1_agonists.
- Trace_amine wikiPageWikiLink Category:Trace_amines.
- Trace_amine wikiPageWikiLink Chemical_synapse.
- Trace_amine wikiPageWikiLink Depression_(mood).
- Trace_amine wikiPageWikiLink Dopamine.
- Trace_amine wikiPageWikiLink Dopamine_neuron.
- Trace_amine wikiPageWikiLink Histamine.
- Trace_amine wikiPageWikiLink Meta-Octopamine.
- Trace_amine wikiPageWikiLink Meta-Tyramine.
- Trace_amine wikiPageWikiLink Metabolism.
- Trace_amine wikiPageWikiLink Methylphenidate.
- Trace_amine wikiPageWikiLink Monoamine_neurotransmitter.
- Trace_amine wikiPageWikiLink N,N-Dimethyltryptamine.
- Trace_amine wikiPageWikiLink N-Methylphenethylamine.
- Trace_amine wikiPageWikiLink N-Methyltryptamine.
- Trace_amine wikiPageWikiLink N-Methyltyramine.
- Trace_amine wikiPageWikiLink Neuromodulation.
- Trace_amine wikiPageWikiLink Neuromodulators.
- Trace_amine wikiPageWikiLink Neurotransmitter.
- Trace_amine wikiPageWikiLink Noradrenaline.
- Trace_amine wikiPageWikiLink Norepinephrine.
- Trace_amine wikiPageWikiLink Norfenefrine.
- Trace_amine wikiPageWikiLink Octopamine.
- Trace_amine wikiPageWikiLink Para-Octopamine.
- Trace_amine wikiPageWikiLink Para-Tyramine.
- Trace_amine wikiPageWikiLink Pharmacodynamics.
- Trace_amine wikiPageWikiLink Phenethylamine.
- Trace_amine wikiPageWikiLink Phenylethanolamine.
- Trace_amine wikiPageWikiLink Schizophrenia.
- Trace_amine wikiPageWikiLink Serotonin.
- Trace_amine wikiPageWikiLink Synaptic_cleft.
- Trace_amine wikiPageWikiLink Synephrine.
- Trace_amine wikiPageWikiLink TAAR1.
- Trace_amine wikiPageWikiLink TAAR1_agonist.
- Trace_amine wikiPageWikiLink Thyronamine.
- Trace_amine wikiPageWikiLink Trace_amine-associated_receptor.
- Trace_amine wikiPageWikiLink Trace_amine-associated_receptor_1.
- Trace_amine wikiPageWikiLink Tryptamine.
- Trace_amine wikiPageWikiLink Tyramine.
- Trace_amine wikiPageWikiLink Vesicular_monoamine_transporter_2.
- Trace_amine wikiPageWikiLinkText "Trace amine".
- Trace_amine wikiPageWikiLinkText "Trace amine#list".
- Trace_amine wikiPageWikiLinkText "its endogenous analogues".
- Trace_amine wikiPageWikiLinkText "phenethylaminergic trace amines".
- Trace_amine wikiPageWikiLinkText "trace amine neuromodulator".
- Trace_amine wikiPageWikiLinkText "trace amine transmitters".
- Trace_amine wikiPageWikiLinkText "trace amine".
- Trace_amine wikiPageWikiLinkText "trace".
- Trace_amine align "right".
- Trace_amine alt "Chemical structure diagrams".
- Trace_amine biologicalTarget TAAR1.
- Trace_amine biologicalTarget Trace_amine-associated_receptor_1.
- Trace_amine caption "Phenethylamine skeleton".
- Trace_amine caption "Phenethylaminergic trace amines and the catecholamines are derivatives of phenylalanine.".
- Trace_amine hasPhotoCollection Trace_amine.
- Trace_amine header "Human biosynthesis pathway for trace amines and catecholamines".
- Trace_amine meshid "434723.0".
- Trace_amine use "Mood and neuropsychiatric disorders".
- Trace_amine wikiPageUsesTemplate Template:Abbr.
- Trace_amine wikiPageUsesTemplate Template:Amphetamine.
- Trace_amine wikiPageUsesTemplate Template:Anchor.
- Trace_amine wikiPageUsesTemplate Template:Clear.
- Trace_amine wikiPageUsesTemplate Template:Infobox_drug_class.
- Trace_amine wikiPageUsesTemplate Template:Neurotransmitters.
- Trace_amine wikiPageUsesTemplate Template:Phenylalanine_biosynthesis.
- Trace_amine wikiPageUsesTemplate Template:Reflist.
- Trace_amine wikiPageUsesTemplate Template:TAAR_ligands.
- Trace_amine wikiPageUsesTemplate Template:Use_dmy_dates.
- Trace_amine subject Category:Amines.
- Trace_amine subject Category:Amphetamine.
- Trace_amine subject Category:Neurochemistry.
- Trace_amine subject Category:Neurotransmitters.
- Trace_amine subject Category:TAAR1_agonists.
- Trace_amine subject Category:Trace_amines.
- Trace_amine hypernym Group.
- Trace_amine type Band.
- Trace_amine type Biomolecule.
- Trace_amine type Group.
- Trace_amine type Biomolecule.
- Trace_amine type Group.
- Trace_amine type Concept.
- Trace_amine comment "Trace amines are an endogenous group of trace amine associated receptor 1 (TAAR1) agonists – and hence, monoaminergic neuromodulators – that are structurally and metabolically related to classical monoamine neurotransmitters. Compared to the classical monoamines, they are present in trace concentrations. They are distributed heterogeneously throughout the mammalian brain and peripheral nervous tissues and exhibit high rates of metabolism.".
- Trace_amine label "Trace amine".
- Trace_amine sameAs Category:Trace_amine.