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- Tivozanib abstract "Tivozanib (AV-951) is an oral VEGF receptor tyrosine kinase inhibitor. It is undergoing clinical trial investigation for the treatment of renal cell carcinomas. An oral quinoline urea derivative, tivozanib suppresses angiogenesis by being selectively inhibitory against vascular endothelial growth factor. It was developed by AVEO Pharmaceuticals. It is designed to inhibit all three VEGF receptors.Phase III results on advanced renal cell carcinoma suggest a 30% or 3 months improvement in median PFS compared to sorafenib. The Food and Drug Administration's Oncologic Drugs Advisory Committee voted in May 2013 13 to 1 against recommending approval of tivozanib for renal cell carcinoma. The committee felt the drug failed to show a favorable risk-benefit ratio and questioned the equipose of the trial design, which allowed control arm patients who used sorafenib to transition to tivozanib following progression disease but not those on the experimental arm using tivozanib to transition to sorafenib. There was an inferior overall survival rate of the experimental arm versus the control arm in this Phase III study as well. The application was formally rejected by the FDA in June 2013, saying that approval would require additional clinical studies.".
- Tivozanib iupacName "1-{2-Chloro-4-[(6,7-dimethoxyquinolin-4-yl)oxy]phenyl}-3-(5-methylisoxazol-3-yl)urea".
- Tivozanib thumbnail Tivozanib.svg?width=300.
- Tivozanib wikiPageID "27723967".
- Tivozanib wikiPageLength "3625".
- Tivozanib wikiPageOutDegree "19".
- Tivozanib wikiPageRevisionID "668616815".
- Tivozanib wikiPageWikiLink AVEO_Pharmaceuticals.
- Tivozanib wikiPageWikiLink Angiogenesis.
- Tivozanib wikiPageWikiLink Category:Angiogenesis_inhibitors.
- Tivozanib wikiPageWikiLink Category:Experimental_cancer_drugs.
- Tivozanib wikiPageWikiLink Category:Isoxazoles.
- Tivozanib wikiPageWikiLink Category:Quinolines.
- Tivozanib wikiPageWikiLink Category:Receptor_tyrosine_kinase_inhibitors.
- Tivozanib wikiPageWikiLink Food_and_Drug_Administration.
- Tivozanib wikiPageWikiLink New_drug_application.
- Tivozanib wikiPageWikiLink New_drug_application_(FDA).
- Tivozanib wikiPageWikiLink Progression-free_survival.
- Tivozanib wikiPageWikiLink Quinoline.
- Tivozanib wikiPageWikiLink Renal_cell_carcinoma.
- Tivozanib wikiPageWikiLink Sorafenib.
- Tivozanib wikiPageWikiLink Tyrosine_kinase.
- Tivozanib wikiPageWikiLink Urea.
- Tivozanib wikiPageWikiLink VEGF_receptor.
- Tivozanib wikiPageWikiLink VEGF_receptors.
- Tivozanib wikiPageWikiLink Vascular_endothelial_growth_factor.
- Tivozanib wikiPageWikiLinkText "Tivozanib".
- Tivozanib wikiPageWikiLinkText "tivozanib".
- Tivozanib hasPhotoCollection Tivozanib.
- Tivozanib imagefile "Tivozanib.svg".
- Tivozanib imagesize "200".
- Tivozanib iupacname "1".
- Tivozanib othernames "AV-951".
- Tivozanib wikiPageUsesTemplate Template:Chembox.
- Tivozanib wikiPageUsesTemplate Template:Pharma-stub.
- Tivozanib wikiPageUsesTemplate Template:Reflist.
- Tivozanib subject Category:Angiogenesis_inhibitors.
- Tivozanib subject Category:Experimental_cancer_drugs.
- Tivozanib subject Category:Isoxazoles.
- Tivozanib subject Category:Quinolines.
- Tivozanib subject Category:Receptor_tyrosine_kinase_inhibitors.
- Tivozanib hypernym Inhibitor.
- Tivozanib type Article.
- Tivozanib type ChemicalCompound.
- Tivozanib type ChemicalSubstance.
- Tivozanib type Drug.
- Tivozanib type Article.
- Tivozanib type Azole.
- Tivozanib type Chemical.
- Tivozanib type Drug.
- Tivozanib type Heterocycle.
- Tivozanib type Inhibitor.
- Tivozanib type ChemicalObject.
- Tivozanib type Thing.
- Tivozanib type Q11173.
- Tivozanib comment "Tivozanib (AV-951) is an oral VEGF receptor tyrosine kinase inhibitor. It is undergoing clinical trial investigation for the treatment of renal cell carcinomas. An oral quinoline urea derivative, tivozanib suppresses angiogenesis by being selectively inhibitory against vascular endothelial growth factor. It was developed by AVEO Pharmaceuticals.".
- Tivozanib label "Tivozanib".
- Tivozanib sameAs Tivozanib.
- Tivozanib sameAs m.0cc8_6z.
- Tivozanib sameAs Tivozanib.
- Tivozanib sameAs Tivozanib.
- Tivozanib sameAs Q7810457.
- Tivozanib sameAs Q7810457.
- Tivozanib wasDerivedFrom Tivozanib?oldid=668616815.
- Tivozanib depiction Tivozanib.svg.
- Tivozanib isPrimaryTopicOf Tivozanib.