Matches in DBpedia 2015-10 for { <http://dbpedia.org/resource/Renin_inhibitor> ?p ?o }
- Renin_inhibitor abstract "Renin inhibitors are a group of pharmaceutical drugs used primarily in treatment of essential hypertension (high blood pressure).These drugs inhibit the first and rate-limiting step of the renin–angiotensin–aldosterone system (RAAS), namely the conversion of angiotensinogen to angiotensin I.This leads to a totality in absence of Angiotensin II based on the rationale that renin only acts to inhibit this step unlike Angiotensin Converting Enzyme which is also involved in other biochemical reactions. Since the 1970s, scientists have been trying to develop potent inhibitors with acceptable oral bioavailability. The process was difficult and took about three decades. The first and second generations faced problems such as poor bioavailability and lack of potency. Finally, the third generation was discovered. These compounds were nonpeptidic renin inhibitors, had acceptable oral bioavailability and were potent enough for clinical use. The first drug in this class was aliskiren, which received a marketing approval in 2007. As of January 2012, it is the only renin inhibitor on the market.".
- Renin_inhibitor thumbnail Aliskiren.svg?width=300.
- Renin_inhibitor wikiPageExternalLink 21094.php.
- Renin_inhibitor wikiPageID "14778970".
- Renin_inhibitor wikiPageLength "41146".
- Renin_inhibitor wikiPageOutDegree "140".
- Renin_inhibitor wikiPageRevisionID "678196230".
- Renin_inhibitor wikiPageWikiLink ACE_inhibitor.
- Renin_inhibitor wikiPageWikiLink ACE_inhibitors_drug_design.
- Renin_inhibitor wikiPageWikiLink Active_site.
- Renin_inhibitor wikiPageWikiLink Affinity_(pharmacology).
- Renin_inhibitor wikiPageWikiLink Aldosterone.
- Renin_inhibitor wikiPageWikiLink Aliskiren.
- Renin_inhibitor wikiPageWikiLink Amine.
- Renin_inhibitor wikiPageWikiLink Amino_acid.
- Renin_inhibitor wikiPageWikiLink Angiotensin.
- Renin_inhibitor wikiPageWikiLink Angiotensin-converting_enzyme.
- Renin_inhibitor wikiPageWikiLink Angiotensin_I.
- Renin_inhibitor wikiPageWikiLink Angiotensin_II.
- Renin_inhibitor wikiPageWikiLink Angiotensin_II_receptor_antagonist.
- Renin_inhibitor wikiPageWikiLink Angiotensin_II_receptor_type_1.
- Renin_inhibitor wikiPageWikiLink Angiotensin_II_receptor_type_2.
- Renin_inhibitor wikiPageWikiLink Angiotensin_receptor.
- Renin_inhibitor wikiPageWikiLink Angiotensinogen.
- Renin_inhibitor wikiPageWikiLink Arginine.
- Renin_inhibitor wikiPageWikiLink Aromatic.
- Renin_inhibitor wikiPageWikiLink Aromaticity.
- Renin_inhibitor wikiPageWikiLink Aspartate_protease.
- Renin_inhibitor wikiPageWikiLink Aspartic_acid.
- Renin_inhibitor wikiPageWikiLink Aspartic_protease.
- Renin_inhibitor wikiPageWikiLink Beta_blocker.
- Renin_inhibitor wikiPageWikiLink Beta_hairpin.
- Renin_inhibitor wikiPageWikiLink Beta_sheet.
- Renin_inhibitor wikiPageWikiLink Bioavailability.
- Renin_inhibitor wikiPageWikiLink Blood_plasma.
- Renin_inhibitor wikiPageWikiLink Blood_pressure.
- Renin_inhibitor wikiPageWikiLink Carboxylic_acid.
- Renin_inhibitor wikiPageWikiLink Cardiac_output.
- Renin_inhibitor wikiPageWikiLink Cardiovascular_disease.
- Renin_inhibitor wikiPageWikiLink Catalysis.
- Renin_inhibitor wikiPageWikiLink Category:Articles_created_via_the_Article_Wizard.
- Renin_inhibitor wikiPageWikiLink Category:Renin_inhibitors.
- Renin_inhibitor wikiPageWikiLink Cathepsin_D.
- Renin_inhibitor wikiPageWikiLink Chemical_compound.
- Renin_inhibitor wikiPageWikiLink Chemical_decomposition.
- Renin_inhibitor wikiPageWikiLink Chemical_polarity.
- Renin_inhibitor wikiPageWikiLink Chemical_synthesis.
- Renin_inhibitor wikiPageWikiLink Circulatory_system.
- Renin_inhibitor wikiPageWikiLink Clinical_trial.
- Renin_inhibitor wikiPageWikiLink Combination_therapy.
- Renin_inhibitor wikiPageWikiLink Competitive_inhibition.
- Renin_inhibitor wikiPageWikiLink Competitive_inhibitor.
- Renin_inhibitor wikiPageWikiLink Concentration.
- Renin_inhibitor wikiPageWikiLink Crystallography.
- Renin_inhibitor wikiPageWikiLink Decapeptide.
- Renin_inhibitor wikiPageWikiLink Diabetes_mellitus.
- Renin_inhibitor wikiPageWikiLink Discovery_and_development_of_ACE_inhibitors.
- Renin_inhibitor wikiPageWikiLink Discovery_and_development_of_angiotensin_receptor_blockers.
- Renin_inhibitor wikiPageWikiLink Distribution_(pharmacology).
- Renin_inhibitor wikiPageWikiLink Duodenal.
- Renin_inhibitor wikiPageWikiLink Duodenum.
- Renin_inhibitor wikiPageWikiLink End_organ_damage.
- Renin_inhibitor wikiPageWikiLink Enzyme.
- Renin_inhibitor wikiPageWikiLink Enzyme_inhibitor.
- Renin_inhibitor wikiPageWikiLink Enzyme_substrate_(biology).
- Renin_inhibitor wikiPageWikiLink Essential_hypertension.
- Renin_inhibitor wikiPageWikiLink European_Medicines_Agency.
- Renin_inhibitor wikiPageWikiLink Extract.
- Renin_inhibitor wikiPageWikiLink Food_and_Drug_Administration.
- Renin_inhibitor wikiPageWikiLink Functional_selectivity.
- Renin_inhibitor wikiPageWikiLink Glycine.
- Renin_inhibitor wikiPageWikiLink Heart_failure.
- Renin_inhibitor wikiPageWikiLink Homeostasis.
- Renin_inhibitor wikiPageWikiLink Hydrochlorothiazide.
- Renin_inhibitor wikiPageWikiLink Hydrogen_bond.
- Renin_inhibitor wikiPageWikiLink Hydrophile.
- Renin_inhibitor wikiPageWikiLink Hydrophilic.
- Renin_inhibitor wikiPageWikiLink Hydrophobe.
- Renin_inhibitor wikiPageWikiLink Hydrophobic.
- Renin_inhibitor wikiPageWikiLink Hyperkalemia.
- Renin_inhibitor wikiPageWikiLink Hypertension.
- Renin_inhibitor wikiPageWikiLink Hypotension.
- Renin_inhibitor wikiPageWikiLink In_vivo.
- Renin_inhibitor wikiPageWikiLink Jugular_vein.
- Renin_inhibitor wikiPageWikiLink Juxtaglomerular_apparatus.
- Renin_inhibitor wikiPageWikiLink Kidney_disease.
- Renin_inhibitor wikiPageWikiLink Ligand.
- Renin_inhibitor wikiPageWikiLink Ligand_(biochemistry).
- Renin_inhibitor wikiPageWikiLink Lipophilic.
- Renin_inhibitor wikiPageWikiLink Lipophilicity.
- Renin_inhibitor wikiPageWikiLink Marmoset.
- Renin_inhibitor wikiPageWikiLink Methoxy.
- Renin_inhibitor wikiPageWikiLink Microorganism.
- Renin_inhibitor wikiPageWikiLink Molecular_modeling.
- Renin_inhibitor wikiPageWikiLink Molecular_modelling.
- Renin_inhibitor wikiPageWikiLink Monotherapy.
- Renin_inhibitor wikiPageWikiLink N-terminus.
- Renin_inhibitor wikiPageWikiLink Negative_feedback.
- Renin_inhibitor wikiPageWikiLink Parenterally.
- Renin_inhibitor wikiPageWikiLink Pathogenesis.