Matches in DBpedia 2015-10 for { <http://dbpedia.org/resource/Receptor_antagonist> ?p ?o }
- Receptor_antagonist abstract "A receptor antagonist is a type of receptor ligand or drug that blocks or dampens agonist-mediated responses rather than provoking a biological response itself upon binding to a receptor. They are sometimes called blockers; examples include alpha blockers, beta blockers, and calcium channel blockers. In pharmacology, antagonists have affinity but no efficacy for their cognate receptors, and binding will disrupt the interaction and inhibit the function of an agonist or inverse agonist at receptors. Antagonists mediate their effects by binding to the active (orthosteric = right place) site or to allosteric (= other place) sites on receptors, or they may interact at unique binding sites not normally involved in the biological regulation of the receptor's activity. Antagonist activity may be reversible or irreversible depending on the longevity of the antagonist–receptor complex, which, in turn, depends on the nature of antagonist–receptor binding. The majority of drug antagonists achieve their potency by competing with endogenous ligands or substrates at structurally defined binding sites on receptors.".
- Receptor_antagonist thumbnail Antagonist_2.png?width=300.
- Receptor_antagonist wikiPageID "654168".
- Receptor_antagonist wikiPageLength "27881".
- Receptor_antagonist wikiPageOutDegree "94".
- Receptor_antagonist wikiPageRevisionID "678664960".
- Receptor_antagonist wikiPageWikiLink Adrenaline.
- Receptor_antagonist wikiPageWikiLink Adrenergic_receptor.
- Receptor_antagonist wikiPageWikiLink Affinity_(pharmacology).
- Receptor_antagonist wikiPageWikiLink Agonist.
- Receptor_antagonist wikiPageWikiLink Allosteric.
- Receptor_antagonist wikiPageWikiLink Allosteric_regulation.
- Receptor_antagonist wikiPageWikiLink Alpha_adrenergic_receptor.
- Receptor_antagonist wikiPageWikiLink Alpha_blocker.
- Receptor_antagonist wikiPageWikiLink Alzheimers_disease.
- Receptor_antagonist wikiPageWikiLink Analgesic.
- Receptor_antagonist wikiPageWikiLink Antihistamine.
- Receptor_antagonist wikiPageWikiLink Beta_blocker.
- Receptor_antagonist wikiPageWikiLink Binding_affinity.
- Receptor_antagonist wikiPageWikiLink Binding_site.
- Receptor_antagonist wikiPageWikiLink Buprenorphine.
- Receptor_antagonist wikiPageWikiLink Calcium_channel_blocker.
- Receptor_antagonist wikiPageWikiLink Category:Pharmacodynamics.
- Receptor_antagonist wikiPageWikiLink Category:Receptor_antagonists.
- Receptor_antagonist wikiPageWikiLink Category:Signal_transduction.
- Receptor_antagonist wikiPageWikiLink Cell_nucleus.
- Receptor_antagonist wikiPageWikiLink Competitive_antagonist.
- Receptor_antagonist wikiPageWikiLink Covalent_bond.
- Receptor_antagonist wikiPageWikiLink Cyclothiazide.
- Receptor_antagonist wikiPageWikiLink Dose-response_curve.
- Receptor_antagonist wikiPageWikiLink Dose–response_relationship.
- Receptor_antagonist wikiPageWikiLink Drug.
- Receptor_antagonist wikiPageWikiLink EC50.
- Receptor_antagonist wikiPageWikiLink Efficacy.
- Receptor_antagonist wikiPageWikiLink Enzyme_inhibitor.
- Receptor_antagonist wikiPageWikiLink Epinephrine.
- Receptor_antagonist wikiPageWikiLink Functional_Selectivity.
- Receptor_antagonist wikiPageWikiLink Functional_selectivity.
- Receptor_antagonist wikiPageWikiLink Growth_factor_receptor_inhibitor.
- Receptor_antagonist wikiPageWikiLink Histamine.
- Receptor_antagonist wikiPageWikiLink Histamine_H1_receptor.
- Receptor_antagonist wikiPageWikiLink Histamine_antagonist.
- Receptor_antagonist wikiPageWikiLink Hormone.
- Receptor_antagonist wikiPageWikiLink IC50.
- Receptor_antagonist wikiPageWikiLink IL1ra.
- Receptor_antagonist wikiPageWikiLink Interleukin-1.
- Receptor_antagonist wikiPageWikiLink Interleukin_1_family.
- Receptor_antagonist wikiPageWikiLink Interleukin_1_receptor_antagonist.
- Receptor_antagonist wikiPageWikiLink Intracellular_receptor.
- Receptor_antagonist wikiPageWikiLink Intrinsic_activity.
- Receptor_antagonist wikiPageWikiLink Inverse_agonist.
- Receptor_antagonist wikiPageWikiLink Ligand_(biochemistry).
- Receptor_antagonist wikiPageWikiLink Memantine.
- Receptor_antagonist wikiPageWikiLink Metabotropic_glutamate_receptor_1.
- Receptor_antagonist wikiPageWikiLink Methadone.
- Receptor_antagonist wikiPageWikiLink Mitochondrion.
- Receptor_antagonist wikiPageWikiLink antagonist.
- Receptor_antagonist wikiPageWikiLink NMDA_receptor.
- Receptor_antagonist wikiPageWikiLink Non-covalent_interactions.
- Receptor_antagonist wikiPageWikiLink Noncovalent.
- Receptor_antagonist wikiPageWikiLink Noradrenaline.
- Receptor_antagonist wikiPageWikiLink Norepinephrine.
- Receptor_antagonist wikiPageWikiLink Opioid_receptor.
- Receptor_antagonist wikiPageWikiLink Opioid_receptors.
- Receptor_antagonist wikiPageWikiLink Partial_agonist.
- Receptor_antagonist wikiPageWikiLink Pharmacodynamics.
- Receptor_antagonist wikiPageWikiLink Pharmacology.
- Receptor_antagonist wikiPageWikiLink Phenoxybenzamine.
- Receptor_antagonist wikiPageWikiLink Physiological_agonism_and_antagonism.
- Receptor_antagonist wikiPageWikiLink Physiological_antagonists.
- Receptor_antagonist wikiPageWikiLink Potency_(pharmacology).
- Receptor_antagonist wikiPageWikiLink Protein.
- Receptor_antagonist wikiPageWikiLink Receptor-ligand_kinetics.
- Receptor_antagonist wikiPageWikiLink Receptor_(biochemistry).
- Receptor_antagonist wikiPageWikiLink Receptor_reserve.
- Receptor_antagonist wikiPageWikiLink Receptor_theory.
- Receptor_antagonist wikiPageWikiLink Receptor–ligand_kinetics.
- Receptor_antagonist wikiPageWikiLink Schild_regression.
- Receptor_antagonist wikiPageWikiLink Selective_receptor_modulator.
- Receptor_antagonist wikiPageWikiLink Vasodilation.
- Receptor_antagonist wikiPageWikiLink File:Antagonist_2.png.
- Receptor_antagonist wikiPageWikiLinkText "''Antagonists''".
- Receptor_antagonist wikiPageWikiLinkText "Antagonism (pharmacology)".
- Receptor_antagonist wikiPageWikiLinkText "Antagonist".
- Receptor_antagonist wikiPageWikiLinkText "Antagonists".
- Receptor_antagonist wikiPageWikiLinkText "Antagonizing".
- Receptor_antagonist wikiPageWikiLinkText "Neutral antagonists".
- Receptor_antagonist wikiPageWikiLinkText "Non-competitive antagonist".
- Receptor_antagonist wikiPageWikiLinkText "Receptor antagonist".
- Receptor_antagonist wikiPageWikiLinkText "Receptor_antagonist#Reversibility".
- Receptor_antagonist wikiPageWikiLinkText "Receptor_antagonist#Silent_antagonists".
- Receptor_antagonist wikiPageWikiLinkText "Silent antagonist".
- Receptor_antagonist wikiPageWikiLinkText "affinity".
- Receptor_antagonist wikiPageWikiLinkText "antagonise".
- Receptor_antagonist wikiPageWikiLinkText "antagonising".
- Receptor_antagonist wikiPageWikiLinkText "antagonism".
- Receptor_antagonist wikiPageWikiLinkText "antagonist".
- Receptor_antagonist wikiPageWikiLinkText "antagonistic".
- Receptor_antagonist wikiPageWikiLinkText "antagonistically".
- Receptor_antagonist wikiPageWikiLinkText "antagonists".