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- Pitrakinra abstract "Pitrakinra (trade name Aerovant) is a 15-kDa human recombinant protein of wild-type human interleukin-4 (IL-4). It is an IL-4 and IL-13 antagonist that has been studied in phase III clinical trials for the treatment of asthma. Two point mutations on pitrakinra (position 121 mutated from arginine to aspartic acid and position 124 mutated from tyrosine to aspartic acid) confer its ability to block signaling of IL-4 and interleukin-13 (IL-13) by preventing assembly of IL-4 receptor alpha (IL-4Rα) with either IL-2Rγ or IL-13Rα. Upregulation of Th2 cytokines, including IL-4 and IL-13, is thought to be critical for the allergic inflammation associated with atopic diseases such as asthma and eczema. The targets of pitrakinra action are inflammatory cells (dendritic cells, Th2 cells, B cells) and structural cells (smooth muscle, endothelium, epithelium) that express IL-4Rα.The drug has been applied both as a subcutaneous injection and as an inhalation, but the latter formulation proved to be more effective.".
- Pitrakinra atcPrefix "none".
- Pitrakinra iupacName "(L)-methionyl-[121-aspartic acid, 124-aspartic acid]interleukin-4".
- Pitrakinra wikiPageID "13987435".
- Pitrakinra wikiPageLength "7192".
- Pitrakinra wikiPageOutDegree "11".
- Pitrakinra wikiPageRevisionID "678193659".
- Pitrakinra wikiPageWikiLink Allergy.
- Pitrakinra wikiPageWikiLink Asthma.
- Pitrakinra wikiPageWikiLink Atomic_mass_unit.
- Pitrakinra wikiPageWikiLink Category:Antiasthmatic_drugs.
- Pitrakinra wikiPageWikiLink Category:Recombinant_proteins.
- Pitrakinra wikiPageWikiLink Immune_response.
- Pitrakinra wikiPageWikiLink Immune_system.
- Pitrakinra wikiPageWikiLink Interleukin-4_receptor.
- Pitrakinra wikiPageWikiLink KDa.
- Pitrakinra wikiPageWikiLink Phase_III_clinical_trial.
- Pitrakinra wikiPageWikiLink Phases_of_clinical_research.
- Pitrakinra wikiPageWikiLink Recombinant_DNA.
- Pitrakinra wikiPageWikiLink Recombinant_protein.
- Pitrakinra wikiPageWikiLink Subcutaneous_injection.
- Pitrakinra wikiPageWikiLink T_helper_cell.
- Pitrakinra wikiPageWikiLink Th2.
- Pitrakinra wikiPageWikiLinkText "Pitrakinra".
- Pitrakinra wikiPageWikiLinkText "pitrakinra".
- Pitrakinra atcPrefix "none".
- Pitrakinra c "651".
- Pitrakinra chembl "2109159".
- Pitrakinra chemspiderid "NA".
- Pitrakinra h "1054".
- Pitrakinra hasPhotoCollection Pitrakinra.
- Pitrakinra iupacName "(L)-methionyl-[121-aspartic acid, 124-aspartic acid]interleukin-4".
- Pitrakinra legalStatus "Investigational".
- Pitrakinra molecularWeight "15".
- Pitrakinra n "190".
- Pitrakinra o "200".
- Pitrakinra routesOfAdministration "Inhalation,".
- Pitrakinra s "8".
- Pitrakinra tradename "Aerovant".
- Pitrakinra wikiPageUsesTemplate Template:Drugbox.
- Pitrakinra wikiPageUsesTemplate Template:Orphan.
- Pitrakinra wikiPageUsesTemplate Template:Reflist.
- Pitrakinra subject Category:Antiasthmatic_drugs.
- Pitrakinra subject Category:Recombinant_proteins.
- Pitrakinra type Article.
- Pitrakinra type ChemicalSubstance.
- Pitrakinra type Drug.
- Pitrakinra type Article.
- Pitrakinra type Disorder.
- Pitrakinra type Page.
- Pitrakinra type Specialty.
- Pitrakinra type ChemicalObject.
- Pitrakinra type Thing.
- Pitrakinra type Q8386.
- Pitrakinra comment "Pitrakinra (trade name Aerovant) is a 15-kDa human recombinant protein of wild-type human interleukin-4 (IL-4). It is an IL-4 and IL-13 antagonist that has been studied in phase III clinical trials for the treatment of asthma.".
- Pitrakinra label "Pitrakinra".
- Pitrakinra sameAs m.03cq834.
- Pitrakinra sameAs Q7199029.
- Pitrakinra sameAs Q7199029.
- Pitrakinra wasDerivedFrom Pitrakinra?oldid=678193659.
- Pitrakinra isPrimaryTopicOf Pitrakinra.