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- Membrane_androgen_receptor abstract "Membrane androgen receptors (mARs) are a group of G protein-coupled receptors (GPCRs) which bind and are activated by testosterone and/or other androgens. Unlike the androgen receptor (AR), a nuclear receptor which mediates its effects via genomic mechanisms, mARs are cell surface receptors which rapidly alter cell signaling via modulation of intracellular signaling cascades. Known or proposed mARs include GPRC6A and ZIP9.GPRC6A has been found to be involved in testicular function and prostate cancer. mARs have also been found to be expressed in breast cancer cells. Activation of mARs by testosterone has been found to increase skeletal muscle strength, indicating potential anabolic effects. mARs have also been implicated in the antigonadotropic effects of androgens. 3α-Androstanediol, an active metabolite of dihydrotestosterone (DHT) and a weak androgen as well as a neurosteroid via acting as a positive allosteric modulator of the GABAA receptor, rapidly influences sexual receptivity and behavior in animals, an effect that is GABAA receptor-dependent.".
- Membrane_androgen_receptor wikiPageID "47502870".
- Membrane_androgen_receptor wikiPageLength "4058".
- Membrane_androgen_receptor wikiPageOutDegree "31".
- Membrane_androgen_receptor wikiPageRevisionID "675692687".
- Membrane_androgen_receptor wikiPageWikiLink 3α-Androstanediol.
- Membrane_androgen_receptor wikiPageWikiLink Active_metabolite.
- Membrane_androgen_receptor wikiPageWikiLink Allosteric_modulator.
- Membrane_androgen_receptor wikiPageWikiLink Anabolic_steroid.
- Membrane_androgen_receptor wikiPageWikiLink Androgen.
- Membrane_androgen_receptor wikiPageWikiLink Androgen_receptor.
- Membrane_androgen_receptor wikiPageWikiLink Antigonadotropic.
- Membrane_androgen_receptor wikiPageWikiLink Antigonadotropin.
- Membrane_androgen_receptor wikiPageWikiLink Breast_cancer.
- Membrane_androgen_receptor wikiPageWikiLink Category:Androgens.
- Membrane_androgen_receptor wikiPageWikiLink Category:G_protein_coupled_receptors.
- Membrane_androgen_receptor wikiPageWikiLink Category:Human_proteins.
- Membrane_androgen_receptor wikiPageWikiLink Cell_signaling.
- Membrane_androgen_receptor wikiPageWikiLink Cell_surface_receptor.
- Membrane_androgen_receptor wikiPageWikiLink Dihydrotestosterone.
- Membrane_androgen_receptor wikiPageWikiLink Estrous_cycle.
- Membrane_androgen_receptor wikiPageWikiLink GABAA_receptor.
- Membrane_androgen_receptor wikiPageWikiLink GPRC6A.
- Membrane_androgen_receptor wikiPageWikiLink G_protein-coupled_receptor.
- Membrane_androgen_receptor wikiPageWikiLink G_protein–coupled_receptor.
- Membrane_androgen_receptor wikiPageWikiLink Genome.
- Membrane_androgen_receptor wikiPageWikiLink Human_sexual_activity.
- Membrane_androgen_receptor wikiPageWikiLink Intracellular.
- Membrane_androgen_receptor wikiPageWikiLink Membrane_steroid_receptor.
- Membrane_androgen_receptor wikiPageWikiLink Neuroactive_steroid.
- Membrane_androgen_receptor wikiPageWikiLink Neurosteroid.
- Membrane_androgen_receptor wikiPageWikiLink Nuclear_receptor.
- Membrane_androgen_receptor wikiPageWikiLink Positive_allosteric_modulator.
- Membrane_androgen_receptor wikiPageWikiLink Prostate_cancer.
- Membrane_androgen_receptor wikiPageWikiLink SLC30A9.
- Membrane_androgen_receptor wikiPageWikiLink Sexual_behavior.
- Membrane_androgen_receptor wikiPageWikiLink Sexual_receptivity.
- Membrane_androgen_receptor wikiPageWikiLink Signal_transduction.
- Membrane_androgen_receptor wikiPageWikiLink Skeletal_muscle.
- Membrane_androgen_receptor wikiPageWikiLink Testicle.
- Membrane_androgen_receptor wikiPageWikiLink Testosterone.
- Membrane_androgen_receptor wikiPageWikiLinkText "Membrane androgen receptor".
- Membrane_androgen_receptor wikiPageWikiLinkText "membrane androgen receptor".
- Membrane_androgen_receptor hasPhotoCollection Membrane_androgen_receptor.
- Membrane_androgen_receptor wikiPageUsesTemplate Template:Androgenics.
- Membrane_androgen_receptor wikiPageUsesTemplate Template:G_protein-coupled_receptors.
- Membrane_androgen_receptor wikiPageUsesTemplate Template:Receptor-stub.
- Membrane_androgen_receptor wikiPageUsesTemplate Template:Reflist.
- Membrane_androgen_receptor subject Category:Androgens.
- Membrane_androgen_receptor subject Category:G_protein_coupled_receptors.
- Membrane_androgen_receptor subject Category:Human_proteins.
- Membrane_androgen_receptor hypernym Group.
- Membrane_androgen_receptor type Band.
- Membrane_androgen_receptor comment "Membrane androgen receptors (mARs) are a group of G protein-coupled receptors (GPCRs) which bind and are activated by testosterone and/or other androgens. Unlike the androgen receptor (AR), a nuclear receptor which mediates its effects via genomic mechanisms, mARs are cell surface receptors which rapidly alter cell signaling via modulation of intracellular signaling cascades.".
- Membrane_androgen_receptor label "Membrane androgen receptor".
- Membrane_androgen_receptor wasDerivedFrom Membrane_androgen_receptor?oldid=675692687.
- Membrane_androgen_receptor isPrimaryTopicOf Membrane_androgen_receptor.