Matches in DBpedia 2015-10 for { <http://dbpedia.org/resource/GABAA_receptor_positive_allosteric_modulator> ?p ?o }
- GABAA_receptor_positive_allosteric_modulator abstract "In pharmacology, GABAA receptor positive allosteric modulators are positive allosteric modulator (PAM) molecules that increase the activity of the GABAA receptor protein in the vertebrate central nervous system. Unlike GABAA receptor agonists, GABAA PAMs do not bind at the same active site as the γ-Aminobutyric acid (GABA) neurotransmitter molecule: PAMs affect the receptor by binding at a different site on the protein. This is called allosteric modulation.GABA is a major inhibitory neurotransmitter in the Central nervous system. By binding it triggers the GABAA receptor to open its chloride channel to allow chlorine ions into the neuron, making the cell hyperpolarized and less likely to fire. GABAA PAMs bind to a different site and increase the effect of GABA by making the channel open more frequently or for longer when GABA binds. However, they do not have an effect if GABA or another agonist is not present.In psychopharmacology, GABAA receptor PAMs used as drugs have mainly sedative and anxiolytic effects. Examples of GABAA PAMs include alcohol (ethanol), benzodiazepines such as diazepam (Valium) and alprazolam (Xanax), Z-drugs such as zolpidem (Ambien), and the barbiturate drugs.".
- GABAA_receptor_positive_allosteric_modulator thumbnail Gamma-Aminobuttersäure_-_gamma-aminobutyric_acid.svg?width=300.
- GABAA_receptor_positive_allosteric_modulator wikiPageID "41069253".
- GABAA_receptor_positive_allosteric_modulator wikiPageLength "28773".
- GABAA_receptor_positive_allosteric_modulator wikiPageOutDegree "122".
- GABAA_receptor_positive_allosteric_modulator wikiPageRevisionID "683189212".
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Action_potential.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Active_site.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Adinazolam.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Adolf_von_Baeyer.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Agonist.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Alcohol.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Alcoholic_beverage.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Alkyne.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Alkynyl.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Allopregnanolone.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Allosteric_modulator.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Allosteric_regulation.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Alprazolam.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Analgesia.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Analgesic.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Anticonvulsant.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Anxiety.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Anxiolytic.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Barbiturate.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Barbiturates.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Barbituric_acid.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Benzodiazepine.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Benzodiazepines.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Butabarbital.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Category:Drug_discovery.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Category:Receptor_modulators.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Central_nervous_system.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Chlordiazepoxide.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Chloride.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Corticosterone.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Dehydroepiandrosterone.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Depression_(physiology).
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Diazepam.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Diethyl_malonate.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Dissociation_constant.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Dosage_form.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Electrophile.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Electrophilic.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Ephedrine.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Epilepsy.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Epileptic.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Ethanol.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Exogenously.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Exogeny.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink GABA.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink GABAA_receptor.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink GABA_agonist.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink GABA_antagonist.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink GABA_receptor.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink GABA_receptor_agonist.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink GABA_receptor_antagonist.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Gamma-Aminobutyric_acid.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Hans_Selye.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Hydroxylation.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Hyperalgesia.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Hyperalgesic.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Hyperpolarization_(biology).
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Hypnotic.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Hypnotics.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Inflammation.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Intrathecal.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Intrathecal_administration.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Ion_channel.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Knoevenagel_condensation.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Lipophilic.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Lipophilicity.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Malonic_acid.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Methionine.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Muscimol.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink NMDA_receptor.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Neuroactive_steroid.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Neuroactive_steroids.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Neurological_disorder.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Neurological_disorders.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Neuron.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Neuropathic.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Neurosteroids.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Neurotransmitter.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Nonbenzodiazepine.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Pathophysiology.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Pentamer.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Pentameric.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Pentobarbital.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Periaqueductal_gray.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Peripheral_nervous_system.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Peripheral_neuropathy.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Pharmacology.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Phenobarbital.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Positive_allosteric_modulator.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Pregnenolone.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Progesterone.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Progesterone_receptor.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Psychiatric.
- GABAA_receptor_positive_allosteric_modulator wikiPageWikiLink Psychiatry.