Matches in DBpedia 2015-10 for { <http://dbpedia.org/resource/Discovery_and_development_of_antiandrogens> ?p ?o }
- Discovery_and_development_of_antiandrogens abstract "In the 1960s, the first antiandrogen, or androgen antagonist, was discovered. Antiandrogens antagonise the androgen receptor (AR) and thereby block the biological effects of testosterone and dihydrotestosterone (DHT). Antiandrogens are important for men with hormonally responsive diseases like prostate cancer, benign prostatic hyperplasia (BHP), acne, seborrhea, hirsutism and androgen alopecia. Antiandrogens are mainly used for the treatment of prostate diseases. Research from 2010 suggests that ARs could be linked to the disease progression of triple-negative breast cancer and that antiandrogens can potentially be used to treat it.As of 2010 antiandrogens are small molecules and can be either steroidal or nonsteroidal depending on ligand chemistry. Steroidal antiandrogens share a similar steroid structure, while nonsteroidal antiandrogens may have structurally distinctive pharmacophores. Only a limited number of compounds are available for clinical use despite the fact that a very large variety of antiandrogen compounds have been discovered and researched.".
- Discovery_and_development_of_antiandrogens thumbnail Androgen_receptor.png?width=300.
- Discovery_and_development_of_antiandrogens wikiPageExternalLink androgendb.mcgill.ca.
- Discovery_and_development_of_antiandrogens wikiPageID "32986449".
- Discovery_and_development_of_antiandrogens wikiPageLength "41368".
- Discovery_and_development_of_antiandrogens wikiPageOutDegree "193".
- Discovery_and_development_of_antiandrogens wikiPageRevisionID "679687610".
- Discovery_and_development_of_antiandrogens wikiPageWikiLink 5-alpha_reductase.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Abiraterone_acetate.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Ablation.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Acetate.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Acetyl.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Acne_vulgaris.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Agonist.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Alkene.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Alopecia_areata.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Amino_acid.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Androgen.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Androgen_receptor.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Anilide.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Aniline.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Antiandrogen.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Antiandrogen_withdrawal_syndrome.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Apalutamide.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Apoptosis.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Arene_substitution_pattern.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Arene_substitution_patterns.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Aromaticity.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Atraric_acid.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Atrophy.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink BMS-641988.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Benign_prostatic_hyperplasia.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Bicalutamide.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Biochemistry.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Biopsy.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Blood–brain_barrier.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Bristol-Myers_Squibb.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Butanol.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink C-terminus.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink CH5137291.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Carbonyl.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Castration.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Category:Antiandrogens.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Category:Articles_created_via_the_Article_Wizard.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Category:Cancer_research.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Cell_culture.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Central_nervous_system.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Charles_Brenton_Huggins.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Chemical_library.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Chirality.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Chlorine.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Chugai_Pharmaceutical_Co..
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Circular_dichroism.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Clinic.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Clinical_trial.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Coactivator_(genetics).
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Cofactor_(biochemistry).
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Conformational_change.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Conformational_isomerism.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Cyanide.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Cyproterone.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Cyproterone_acetate.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Cytoplasm.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Cytosol.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink DNA-binding_domain.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Dihydrotestosterone.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Discovery_and_development_of_antiandrogens.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink EPI-001.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Enantiomer.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Endogeny.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Endogeny_(biology).
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Enzalutamide.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Epileptic_seizure.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Estrogen.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Finasteride.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink First_pass_effect.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Flutamide.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Food_and_Drug_Administration.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink GABAA_receptor.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Galeterone.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Gene.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Gene_expression.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Gonadotropin.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Gonadotropin-releasing_hormone.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Half-life.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Heat_shock_protein.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Hepatotoxicity.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Hirsutism.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Human_gastrointestinal_tract.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Hydantoin.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Hydrogen_bond.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Hydrolysis.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Hyperplasia.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Hypothalamus.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Imidazole.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink In_vitro.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink In_vivo.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink Indole.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink LG105.
- Discovery_and_development_of_antiandrogens wikiPageWikiLink LG120907.