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- Dalcetrapib abstract "Dalcetrapib or JTT-705 is a CETP inhibitor which was being developed by Hoffmann–La Roche until May 2012. The drug was aimed at raising the blood levels of "good cholesterol" (cholesterol carried in HDL particles, aka HDL-C). Prevailing observations indicate that high HDL levels correlate with better overall cardiovascular health, though it remains unclear whether raising HDL levels consequently leads to an increase in cardiovascular health.A 24 week clinical trial showed that dalcetrapib did increase HDL-C levels, supporting the agent's desired effect. Further, the dal-PLAQUE phase IIb trial found evidence of plaque reduction. Plaque reduction is an anticipated observation following an increase in HDL.As of 2010 five phase II trials had started and there was no evidence of the raised blood pressure seen with torcetrapib.dal-VESSEL phase IIb trial found no evidence of flow-mediated dilatation improvement. A 17% increase of Lp-PLA2 mass level was noted. Lp-PLA2 is associated with coronary heart disease and stroke.dal-OUTCOMES phase III trial passed its first interim review in July, 2011, however, development was halted on May 7, 2012 “due to a lack of clinically meaningful efficacy.”.The results of dal-OUTCOMES III were published in November, 2012.".
- Dalcetrapib iupacName "S-[2-({[1-(2-ethylbutyl)cyclohexyl]carbonyl}amino)phenyl] 2-methylpropanethioate".
- Dalcetrapib thumbnail JTT-705_structure.png?width=300.
- Dalcetrapib wikiPageID "20783559".
- Dalcetrapib wikiPageLength "6987".
- Dalcetrapib wikiPageOutDegree "13".
- Dalcetrapib wikiPageRevisionID "678207011".
- Dalcetrapib wikiPageWikiLink Atheroma.
- Dalcetrapib wikiPageWikiLink CETP_inhibitor.
- Dalcetrapib wikiPageWikiLink Category:Anilides.
- Dalcetrapib wikiPageWikiLink Category:Hoffmann-La_Roche.
- Dalcetrapib wikiPageWikiLink Category:Thioesters.
- Dalcetrapib wikiPageWikiLink Clinical_trial.
- Dalcetrapib wikiPageWikiLink Coronary_artery_disease.
- Dalcetrapib wikiPageWikiLink Coronary_heart_disease.
- Dalcetrapib wikiPageWikiLink Good_cholesterol.
- Dalcetrapib wikiPageWikiLink High-density_lipoprotein.
- Dalcetrapib wikiPageWikiLink Hoffmann-La_Roche.
- Dalcetrapib wikiPageWikiLink Hoffmann–La_Roche.
- Dalcetrapib wikiPageWikiLink Lipoprotein-associated_phospholipase_A2.
- Dalcetrapib wikiPageWikiLink Stroke.
- Dalcetrapib wikiPageWikiLink Torcetrapib.
- Dalcetrapib wikiPageWikiLinkText "Dalcetrapib".
- Dalcetrapib wikiPageWikiLinkText "dalcetrapib".
- Dalcetrapib hasPhotoCollection Dalcetrapib.
- Dalcetrapib imagefile "JTT-705_structure.png".
- Dalcetrapib iupacname "S-[2-phenyl] 2-methylpropanethioate".
- Dalcetrapib wikiPageUsesTemplate Template:As_of.
- Dalcetrapib wikiPageUsesTemplate Template:Chembox.
- Dalcetrapib wikiPageUsesTemplate Template:Citation_needed.
- Dalcetrapib wikiPageUsesTemplate Template:Lipid_modifying_agents.
- Dalcetrapib wikiPageUsesTemplate Template:Reflist.
- Dalcetrapib subject Category:Anilides.
- Dalcetrapib subject Category:Hoffmann-La_Roche.
- Dalcetrapib subject Category:Thioesters.
- Dalcetrapib hypernym Inhibitor.
- Dalcetrapib type Article.
- Dalcetrapib type ChemicalCompound.
- Dalcetrapib type ChemicalSubstance.
- Dalcetrapib type Company.
- Dalcetrapib type Group.
- Dalcetrapib type Article.
- Dalcetrapib type Company.
- Dalcetrapib type Group.
- Dalcetrapib type Thioester.
- Dalcetrapib type ChemicalObject.
- Dalcetrapib type Thing.
- Dalcetrapib type Q11173.
- Dalcetrapib comment "Dalcetrapib or JTT-705 is a CETP inhibitor which was being developed by Hoffmann–La Roche until May 2012. The drug was aimed at raising the blood levels of "good cholesterol" (cholesterol carried in HDL particles, aka HDL-C).".
- Dalcetrapib label "Dalcetrapib".
- Dalcetrapib sameAs m.052_hrf.
- Dalcetrapib sameAs Dalcetrapib.
- Dalcetrapib sameAs Dalcetrapib.
- Dalcetrapib sameAs Q5210285.
- Dalcetrapib sameAs Q5210285.
- Dalcetrapib wasDerivedFrom Dalcetrapib?oldid=678207011.
- Dalcetrapib depiction JTT-705_structure.png.
- Dalcetrapib isPrimaryTopicOf Dalcetrapib.