Matches in DBpedia 2015-10 for { <http://dbpedia.org/resource/CCR5_receptor_antagonist> ?p ?o }
- CCR5_receptor_antagonist abstract "CCR5 receptor antagonists are a class of small molecules that antagonize the CCR5 receptor. The C-C motif chemokine receptor CCR5 is involved in the process by which HIV, the virus that causes AIDS, enters cells. Hence antagonists of this receptor are entry inhibitors and have potential therapeutic applications in the treatment of HIV infections.The life cycle of the HIV presents potential targets for drug therapy, one of them being the viral entry pathway. The C-C motif chemokine receptors CCR5 and CXCR4 are the main chemokine receptors involved in the HIV entry process. These receptors belong to the seven transmembrane G-protein-coupled receptor (GPCR) family and are predominantly expressed on human T-cells, dendritic cells and macrophages, Langerhans cells. They play an important role as co-receptors that HIV type 1 (HIV-1) uses to attach to cells before viral fusion and entry into host cells. HIV isolates can be divided into R5 and X4 strains. R5 strain is when the virus uses the co-receptor CCR5 and X4 strain is when it uses CXCR4. The location of CCR5 receptors at the cell surface, both large and small molecules have the potential to interfere with the CCR5-viral interaction and inhibit viral entry into human cells.".
- CCR5_receptor_antagonist thumbnail HIV_attachment.gif?width=300.
- CCR5_receptor_antagonist wikiPageID "24643329".
- CCR5_receptor_antagonist wikiPageLength "31855".
- CCR5_receptor_antagonist wikiPageOutDegree "112".
- CCR5_receptor_antagonist wikiPageRevisionID "680850456".
- CCR5_receptor_antagonist wikiPageWikiLink AIDS.
- CCR5_receptor_antagonist wikiPageWikiLink Active_compound.
- CCR5_receptor_antagonist wikiPageWikiLink Allosteric.
- CCR5_receptor_antagonist wikiPageWikiLink Allosteric_regulation.
- CCR5_receptor_antagonist wikiPageWikiLink Antiviral_drug.
- CCR5_receptor_antagonist wikiPageWikiLink Aplaviroc.
- CCR5_receptor_antagonist wikiPageWikiLink AstraZeneca.
- CCR5_receptor_antagonist wikiPageWikiLink Autoimmune.
- CCR5_receptor_antagonist wikiPageWikiLink Autoimmunity.
- CCR5_receptor_antagonist wikiPageWikiLink Benzamide.
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- CCR5_receptor_antagonist wikiPageWikiLink Dendritic_cells.
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- CCR5_receptor_antagonist wikiPageWikiLink Discovery_and_development_of_non-nucleoside_reverse_transcriptase_inhibitors.
- CCR5_receptor_antagonist wikiPageWikiLink Discovery_and_development_of_nucleoside_and_nucleotide_reverse-transcriptase_inhibitors.
- CCR5_receptor_antagonist wikiPageWikiLink Electrostatic.
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- CCR5_receptor_antagonist wikiPageWikiLink Enantiomer.
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- CCR5_receptor_antagonist wikiPageWikiLink GPCR.
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- CCR5_receptor_antagonist wikiPageWikiLink Glutamic_acid.
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- CCR5_receptor_antagonist wikiPageWikiLink Phases_of_clinical_research.
- CCR5_receptor_antagonist wikiPageWikiLink Phenylalanine.
- CCR5_receptor_antagonist wikiPageWikiLink Piperazine.
- CCR5_receptor_antagonist wikiPageWikiLink Piperidine.
- CCR5_receptor_antagonist wikiPageWikiLink QT_interval.
- CCR5_receptor_antagonist wikiPageWikiLink Receptor_(biochemistry).
- CCR5_receptor_antagonist wikiPageWikiLink Receptor_antagonist.
- CCR5_receptor_antagonist wikiPageWikiLink Schering-Plough.
- CCR5_receptor_antagonist wikiPageWikiLink Small_molecule.